Total synthesis of ionomycin using ring-opening strategies

Org Lett. 2002 May 30;4(11):1879-82. doi: 10.1021/ol025872f.

Abstract

[structure: see text] The total synthesis of the polyether antibiotic ionomycin, a calcium ionophore, is described. The synthesis demonstrates the utility of ring-opening methodologies as applied to the synthesis of polypropionate and deoxypolypropionate subunits, which are found in two of the four fragments in the synthesis.

MeSH terms

  • Aldehydes / chemistry
  • Anti-Bacterial Agents / chemical synthesis*
  • Calcium / chemistry
  • Hydroxylation
  • Indicators and Reagents
  • Ionomycin / chemical synthesis*
  • Ozone / chemistry
  • Stereoisomerism

Substances

  • Aldehydes
  • Anti-Bacterial Agents
  • Indicators and Reagents
  • Ionomycin
  • Ozone
  • Calcium