3-[123I]Iodo-L-alpha-methyl tyrosine transport into human fibroblasts and comparison with Ewing's sarcoma cells

Nucl Med Biol. 2002 May;29(4):483-90. doi: 10.1016/s0969-8051(02)00291-3.

Abstract

The cellular transport systems and the transport kinetics of [123I]IMT uptake into non-malignant extracranial cells were characterized for the first time. Human fibroblasts were chosen as non-malignant extracranial cells as they are found ubiquitous in the body. [123I]IMT is exclusively transported into fibroblasts via the sodium independent system L. An apparent Michaelis constant K(m) = 116.2 +/- 18.9 microM and a maximum transport velocity V(max) = 191.6 +/- 13.9 pmol x (10(6) cells)(-1) x min(-1) were calculated for the sodium-independent transport. These results were compared with those determined in two malignantly transformed extracranial cell lines, the human Ewing's sarcoma cell lines VH-64 and CADO-ES-1.

Publication types

  • Comparative Study

MeSH terms

  • Bone Neoplasms / diagnostic imaging
  • Bone Neoplasms / metabolism*
  • Cell Line
  • Fibroblasts / diagnostic imaging
  • Fibroblasts / metabolism*
  • Humans
  • Methyltyrosines / pharmacokinetics*
  • Radionuclide Imaging
  • Radiopharmaceuticals / pharmacokinetics
  • Reproducibility of Results
  • Sarcoma, Ewing / diagnostic imaging
  • Sarcoma, Ewing / metabolism*
  • Sensitivity and Specificity
  • Sodium / pharmacokinetics

Substances

  • Methyltyrosines
  • Radiopharmaceuticals
  • Sodium
  • 3-iodo-alpha-methyltyrosine