Human nongastric H+-K+-ATPase: transport properties of ATP1al1 assembled with different beta-subunits

Am J Physiol Cell Physiol. 2002 Jul;283(1):C305-14. doi: 10.1152/ajpcell.00590.2001.

Abstract

To investigate whether nongastric H+-K+-ATPases transport Na+ in exchange for K+ and whether different beta-isoforms influence their transport properties, we compared the functional properties of the catalytic subunit of human nongastric H+-K+-ATPase, ATP1al1 (AL1), and of the Na+-K+-ATPase alpha1-subunit (alpha1) expressed in Xenopus oocytes, with different beta-subunits. Our results show that betaHK and beta1-NK can produce functional AL1/beta complexes at the oocyte cell surface that, in contrast to alpha1/beta1 NK and alpha1/betaHK complexes, exhibit a similar apparent K+ affinity. Similar to Na+-K+-ATPase, AL1/beta complexes are able to decrease intracellular Na+ concentrations in Na+-loaded oocytes, and their K+ transport depends on intra- and extracellular Na+ concentrations. Finally, controlled trypsinolysis reveals that beta-isoforms influence the protease sensitivity of AL1 and alpha1 and that AL1/beta complexes, similar to the Na+-K+-ATPase, can undergo distinct K+-Na+- and ouabain-dependent conformational changes. These results provide new evidence that the human nongastric H+-K+-ATPase interacts with and transports Na+ in exchange for K+ and that beta-isoforms have a distinct effect on the overall structural integrity of AL1 but influence its transport properties less than those of the Na+-K+-ATPase alpha-subunit.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Biological Transport / physiology
  • Cell Membrane / metabolism
  • Enzyme Activation / drug effects
  • Enzyme Inhibitors / pharmacology
  • H(+)-K(+)-Exchanging ATPase / chemistry
  • H(+)-K(+)-Exchanging ATPase / metabolism*
  • Humans
  • Isoenzymes / metabolism
  • Ligands
  • Molecular Conformation
  • Oocytes
  • Ouabain / pharmacology
  • Peptide Hydrolases / metabolism
  • Potassium / pharmacology
  • Protein Processing, Post-Translational*
  • Sodium-Potassium-Exchanging ATPase / chemistry
  • Sodium-Potassium-Exchanging ATPase / drug effects
  • Sodium-Potassium-Exchanging ATPase / metabolism*
  • Xenopus

Substances

  • Enzyme Inhibitors
  • Isoenzymes
  • Ligands
  • Ouabain
  • Peptide Hydrolases
  • ATP12A protein, human
  • H(+)-K(+)-Exchanging ATPase
  • Sodium-Potassium-Exchanging ATPase
  • Potassium