Dominant regulation of interendothelial cell gap formation by calcium-inhibited type 6 adenylyl cyclase

J Cell Biol. 2002 Jun 24;157(7):1267-78. doi: 10.1083/jcb.200204022. Epub 2002 Jun 24.

Abstract

Acute transitions in cytosolic calcium ([Ca2+]i) through store-operated calcium entry channels catalyze interendothelial cell gap formation that increases permeability. However, the rise in [Ca2+]i only disrupts barrier function in the absence of a rise in cAMP. Discovery that type 6 adenylyl cyclase (AC6; EC 4.6.6.1) is inhibited by calcium entry through store-operated calcium entry pathways provided a plausible explanation for how inflammatory [Ca2+]i mediators may decrease cAMP necessary for endothelial cell gap formation. [Ca2+]i mediators only modestly decrease global cAMP concentrations and thus, to date, the physiological role of AC6 is unresolved. Present studies used an adenoviral construct that expresses the calcium-stimulated AC8 to convert normal calcium inhibition into stimulation of cAMP, within physiologically relevant concentration ranges. Thrombin stimulated a dose-dependent [Ca2+]i rise in both pulmonary artery (PAECs) and microvascular (PMVEC) endothelial cells, and promoted intercellular gap formation in both cell types. In PAECs, gap formation was progressive over 2 h, whereas in PMVECs, gap formation was rapid (within 10 min) and gaps resealed within 2 h. Expression of AC8 resulted in a modest calcium stimulation of cAMP, which virtually abolished thrombin-induced gap formation in PMVECs. Findings provide the first direct evidence that calcium inhibition of AC6 is essential for endothelial gap formation.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenoviridae
  • Adenylyl Cyclases / metabolism*
  • Adenylyl Cyclases / physiology
  • Calcium / metabolism*
  • Calcium / pharmacology
  • Cell Communication
  • Cells, Cultured
  • Cyclic AMP / metabolism
  • Cytosol / chemistry
  • Endothelium / cytology*
  • Endothelium / ultrastructure
  • Endothelium, Vascular / cytology
  • Endothelium, Vascular / drug effects
  • Gap Junctions / drug effects
  • Gap Junctions / metabolism*
  • Gap Junctions / ultrastructure
  • Gene Expression Regulation / genetics*
  • Hemostatics / pharmacology
  • Lung / blood supply
  • Pulmonary Artery / cytology
  • Signal Transduction / drug effects
  • Thrombin / pharmacology
  • Time Factors

Substances

  • Hemostatics
  • Cyclic AMP
  • Thrombin
  • Adenylyl Cyclases
  • adenylyl cyclase 6
  • adenylyl cyclase 8
  • Calcium