Snail induction of epithelial to mesenchymal transition in tumor cells is accompanied by MUC1 repression and ZEB1 expression

J Biol Chem. 2002 Oct 18;277(42):39209-16. doi: 10.1074/jbc.M206400200. Epub 2002 Aug 2.

Abstract

E-cadherin protein plays a key role in the establishment and maintenance of adherent junctions. Recent evidence implicates the transcription factor Snail in the blockage of E-cadherin expression in fibroblasts and some epithelial tumor cells through direct binding to three E-boxes in the E-cadherin promoter. Transfection of Snail into epithelial cells leads to a more fibroblastic phenotype. Cells expressing Snail presented a scattered flattened phenotype with low intercellular contacts. Other epithelial markers like Cytokeratin 18 or MUC1 were also repressed. The effects of Snail on MUC1 transcription were mediated by two E-boxes present in the proximal promoter. Snail also induced expression of the mesenchymal markers fibronectin and LEF1 and the transcription repressor ZEB1. ZEB1 and Snail had a similar pattern of expression in epithelial cell lines, and both were induced by overexpression of ILK1, a kinase that causes the loss of E-cadherin and the acquisition of a fibroblastic phenotype. Snail overexpression in several cell lines raised ZEB1 RNA levels and increased the activity of ZEB1 promoter. ZEB1 could also repress E-cadherin and MUC1 promoters but less strongly than Snail. However, since ZEB1 expression persisted after Snail was down-regulated, ZEB1 may regulate epithelial genes in several tumor cell lines.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Blotting, Northern
  • Blotting, Western
  • Cell Line
  • Cell Nucleus / metabolism
  • Cloning, Molecular
  • DNA / metabolism
  • DNA, Complementary / metabolism
  • DNA-Binding Proteins / metabolism*
  • Dogs
  • Down-Regulation
  • Epithelial Cells / metabolism*
  • Fibroblasts / metabolism
  • Humans
  • Keratins / metabolism
  • Mesoderm / metabolism*
  • Mice
  • Microscopy, Electron
  • Mucin-1 / metabolism*
  • Phenotype
  • Promoter Regions, Genetic
  • Protein Binding
  • RNA / metabolism
  • Repressor Proteins / metabolism*
  • Reverse Transcriptase Polymerase Chain Reaction
  • Snail Family Transcription Factors
  • Tetracycline / pharmacology
  • Transcription Factors / metabolism*
  • Transcription, Genetic
  • Transfection
  • Tumor Cells, Cultured
  • Up-Regulation

Substances

  • DNA, Complementary
  • DNA-Binding Proteins
  • Mucin-1
  • Repressor Proteins
  • Snail Family Transcription Factors
  • Transcription Factors
  • RNA
  • Keratins
  • DNA
  • Tetracycline