Synthesis and antiinflammatory activity of novel 3-(2,3-dimethyl-1-phenyl-4-pyrazolon-5-yl)-4-thiazolidones

Boll Chim Farm. 2002 May-Jun;141(3):197-201.

Abstract

New 3-(2,3-dimethyl-1-phenyl-4-pyrazolon-5-yl)-4-thiazolidones were synthesized. The structure of substances was supported by UV- and 1H-NMR spectra. Some compounds were tested in vivo for their antiinflammatory activity. Were confirmed previous results about structure-activity relationships.

MeSH terms

  • Animals
  • Anti-Inflammatory Agents, Non-Steroidal / chemical synthesis*
  • Anti-Inflammatory Agents, Non-Steroidal / pharmacology*
  • Edema / chemically induced
  • Edema / prevention & control
  • Female
  • Indicators and Reagents
  • Magnetic Resonance Spectroscopy
  • Male
  • Rats
  • Spectrophotometry, Ultraviolet
  • Thiazoles / chemical synthesis*
  • Thiazoles / pharmacology*

Substances

  • Anti-Inflammatory Agents, Non-Steroidal
  • Indicators and Reagents
  • Thiazoles