Poly-L-arginine synergizes with oligodeoxynucleotides containing CpG-motifs (CpG-ODN) for enhanced and prolonged immune responses and prevents the CpG-ODN-induced systemic release of pro-inflammatory cytokines

Vaccine. 2002 Oct 4;20(29-30):3498-508. doi: 10.1016/s0264-410x(02)00343-2.

Abstract

This study describes an entirely synthetic vaccine composed of antigenic peptides (T cell epitopes), oligodeoxynucleotides containing CpG-motifs (CpG-ODN) and poly-L-arginine (pR). CpG-ODN are known to be potent inducers of predominantly type 1-like immune responses, while polycationic amino acids, like pR, facilitate the uptake of antigens into antigen presenting cells (APCs). We demonstrate that the application of peptides and pR/CpG-ODN results in strongly enhanced peptide-specific immune responses as compared to the application of peptides with either of the immunomodulators alone. High numbers of antigen-specific T cells can be observed even after only one injection of the vaccine for a remarkably long period of time (at least 372 days). Furthermore, the potentially harmful systemic release of pro-inflammatory cytokines induced upon injection of CpG-ODN is inhibited. Thus, the combined application of CpG-ODN and pR may represent a novel vaccine strategy in humans.

MeSH terms

  • Adjuvants, Immunologic / pharmacology*
  • Animals
  • Cytokines / metabolism*
  • Drug Synergism
  • Female
  • Mice
  • Mice, Inbred C57BL
  • Mice, Inbred DBA
  • Oligodeoxyribonucleotides / pharmacology*
  • Ovalbumin / immunology
  • Peptide Fragments / immunology
  • Peptides / pharmacology*
  • Static Electricity
  • T-Lymphocytes / immunology
  • Vaccination
  • Vaccines, Synthetic / immunology*

Substances

  • Adjuvants, Immunologic
  • CPG-oligonucleotide
  • Cytokines
  • Oligodeoxyribonucleotides
  • Peptide Fragments
  • Peptides
  • Vaccines, Synthetic
  • polyarginine
  • Ovalbumin