Enzymatic oxidation and reduction of C19-delta5-3beta-hydroxysteroids by hepatic microsomes. IV. Induction of DHA hydroxylases and aminopyrine N-demethylase in immature male rats by androgens

Endocrinology. 1975 Mar;96(3):815-9. doi: 10.1210/endo-96-3-815.

Abstract

The capacities of various C19 steroids for prematurely inducing the normal metabolic patterns of rat liver in adulthood (70 days old) have been studied with hepatic microsomes of 42-day-old males castrated on day 24, 30, 32, or 34 of life. Dehydroepiandrosterone 16alpha-hydroxylase activity was significantly reduced (P less than 0.05) by castration during this 10-day interval but the 7alpha- and 7beta-hydroxylases, the N-demethylation of aminopyrine, and cytochrome P-450 concentration were unaffected. Daily administration of testosterone stimulated the DHA 16-alpha- and 17beta-hydroxylases, aminopyrine N-demethylation, and increased the P-450 content, but suppressed the 7alpha-hydroxylase. These effects only appeared with more than 1 week of the continuous treatment. Testosterone was the most active of the androgens studied; dihydrotestosterone (DHT) increased the DHA 16alpha-hydroxylase to a lesser extent, but this steroid and etiocholanolone stimulated DHA 7alpha-hydroxylation; androsterone was totally ineffective. These data suggest that testosterone rather than DHT from pubertal testes plays a significant role in control of hepatic oxidative enzyme activities during puberty.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Age Factors
  • Aminopyrine N-Demethylase / biosynthesis*
  • Androgens / physiology*
  • Androsterone / pharmacology
  • Animals
  • Aryl Hydrocarbon Hydroxylases*
  • Castration
  • Cytochrome P-450 Enzyme System / metabolism
  • Cytochrome P450 Family 2
  • Dehydroepiandrosterone
  • Dihydrotestosterone / pharmacology
  • Enzyme Induction
  • Etiocholanolone / pharmacology
  • Hydroxysteroids / metabolism*
  • Male
  • Microsomes, Liver / enzymology*
  • Mixed Function Oxygenases / biosynthesis*
  • Oxidation-Reduction
  • Rats
  • Steroid 16-alpha-Hydroxylase
  • Stimulation, Chemical
  • Testosterone / pharmacology

Substances

  • Androgens
  • Hydroxysteroids
  • Dihydrotestosterone
  • Testosterone
  • Dehydroepiandrosterone
  • Cytochrome P-450 Enzyme System
  • Etiocholanolone
  • Androsterone
  • Mixed Function Oxygenases
  • Aryl Hydrocarbon Hydroxylases
  • CYP2C11 protein, rat
  • Cytochrome P450 Family 2
  • Steroid 16-alpha-Hydroxylase
  • Aminopyrine N-Demethylase