Reactive oxygen species scavengers attenuate endotoxin-induced impairment of hypoxic pulmonary vasoconstriction in mice

Anesthesiology. 2002 Nov;97(5):1227-33. doi: 10.1097/00000542-200211000-00028.

Abstract

Background: Sepsis and endotoxemia attenuate hypoxic pulmonary vasoconstriction (HPV), thereby impairing systemic oxygenation. Reactive oxygen species (ROS) are implicated in the pathogenesis of sepsis-induced lung injury. The authors investigated whether treatment with scavengers of ROS prevents impairment of HPV in mice challenged with endotoxin.

Methods: The pulmonary vasoconstrictor response to left mainstem bronchus occlusion (LMBO) was studied in anesthetized mice 22 h after an intraperitoneal challenge with saline solution or 10 mg/kg Escherichia coli endotoxin. In some mice, challenge with saline solution or endotoxin was followed after 1 h with intraperitoneal or intratracheal administration of the ROS scavengers N-acetylcysteine or EUK-8. Myeloperoxidase activity and nitric oxide synthase-2 gene expression were measured in lung tissues.

Results: The LMBO increased left pulmonary vascular resistance by 106 +/- 24% in saline-challenged control mice but by only 23 +/- 12% (P < 0.05) in endotoxin-challenged mice. Intraperitoneal administration of N-acetylcysteine or EUK-8 1 h after endotoxin challenge attenuated the endotoxin-induced impairment of HPV (58 +/- 6% and 68 +/- 10%, respectively; both P< 0.05 endotoxin-challenged mice). Intratracheal administration of ROS scavengers 1 h after endotoxin challenge was equally effective but required lower doses than systemic treatment. Administration of the ROS scavengers 22 h after endotoxin challenge did not restore HPV.

Conclusions: Administration of N-acetylcysteine or EUK-8 1 h after endotoxin challenge in mice prevented the impairment of HPV after LMBO. Early therapy with ROS scavengers, either systemically or by inhalation, may provide a means to preserve HPV in sepsis-associated acute lung injury.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Acetylcysteine / pharmacology*
  • Animals
  • Antioxidants / pharmacology*
  • Cell Hypoxia / physiology*
  • Endotoxins / toxicity*
  • Ethylenediamines / pharmacology*
  • Female
  • Male
  • Mice
  • Nitric Oxide Synthase / genetics
  • Nitric Oxide Synthase Type II
  • Organometallic Compounds / pharmacology*
  • Peroxidase / metabolism
  • Pulmonary Circulation / drug effects*
  • RNA, Messenger / analysis
  • Reactive Oxygen Species / metabolism*
  • Respiratory Distress Syndrome / prevention & control
  • Vasoconstriction / drug effects*

Substances

  • Antioxidants
  • Endotoxins
  • Ethylenediamines
  • Organometallic Compounds
  • RNA, Messenger
  • Reactive Oxygen Species
  • N,N'-bis(salicylideneamino)ethane-manganese(II)
  • endotoxin, Escherichia coli
  • Peroxidase
  • Nitric Oxide Synthase
  • Nitric Oxide Synthase Type II
  • Nos2 protein, mouse
  • Acetylcysteine