The role of angiotensin II in hypertension due to adenosine receptors blockade

Eur J Pharmacol. 2002 Nov 29;455(2-3):135-41. doi: 10.1016/s0014-2999(02)02587-6.

Abstract

The renin-angiotensin system may be involved in hypertension induced by adenosine receptors blockade with 1,3-dipropyl-8-sulfophenylxanthine (DPSPX). Contractions of the mesenteric vasculature to angiotensin II, noradrenaline and potassium chloride were studied in DPSPX-induced hypertension. Male Wistar rats received infusions of saline or DPSPX (90 microg kg(-1) h(-1), i.p.) for 3 or 7 days. Blood pressure was determined by the tail-cuff method. On days 3 or 14, concentration-response curves were obtained on mesenteric arteries and veins. Plasma angiotensin II levels, measured by radioimmunoassay, were higher in DPSPX-hypertensive rats. The maximum contractile effect of angiotensin II was lower in vessels from DPSPX-hypertensive rats while that for noradrenaline was higher. Potassium chloride-induced contractions were larger in veins from DPSPX-hypertensive rats but similar in arteries, when compared with control rats. We conclude that raised angiotensin II levels and altered vascular reactivity are consistent with a renin-angiotensin-mediated hypertension.

MeSH terms

  • Angiotensin II / blood
  • Angiotensin II / pharmacology
  • Angiotensin II / physiology*
  • Animals
  • Blood Pressure / drug effects
  • Dose-Response Relationship, Drug
  • Hypertension / physiopathology*
  • In Vitro Techniques
  • Male
  • Mesenteric Arteries / drug effects
  • Mesenteric Arteries / physiopathology
  • Mesenteric Veins / drug effects
  • Mesenteric Veins / physiopathology
  • Norepinephrine / pharmacology
  • Potassium Chloride / pharmacology
  • Purinergic P1 Receptor Antagonists*
  • Rats
  • Rats, Wistar
  • Time Factors
  • Vasoconstriction / drug effects
  • Vasoconstrictor Agents / pharmacology
  • Xanthines / pharmacology

Substances

  • Purinergic P1 Receptor Antagonists
  • Vasoconstrictor Agents
  • Xanthines
  • Angiotensin II
  • Potassium Chloride
  • 1,3-dipropyl-8-(4-sulfophenyl)xanthine
  • Norepinephrine