Topical allopurinol or corticosteroids and acetylcysteine in the early treatment of experimental corneal alkali burns: a pilot study

Eur J Ophthalmol. 2002 Sep-Oct;12(5):366-72. doi: 10.1177/112067210201200504.

Abstract

Purpose: To investigate the effect of topical allopurinol on experimental corneal burns and to compare this to established treatment modalities such as topical prednisolone and acetylcysteine.

Methods: Twenty Wistar rats were randomly assigned to four groups (n=5 each). The groups were controls (normal saline), allopurinol 0.4% eye drops, prednisolone acetate 1% eye drops and acetylcysteine 8% eyedrops. Corneal burn was induced using a 3 mm paper disc soaked in 1N NaOH for 60 seconds. Drops were instilled 6 times per day. In addition, one drop/day ofloxacine was given to prevent secondary infections. Eyes were enucleated 50 hours later and fixed in 4.5% formaldehyde. Three histological levels of each globe were stained with hematoxylin-eosin and examined by two independent masked investigators using a 0 to 4+ inflammatory score. All pair-wise multiple comparison procedures (Student-Newman-Keuls method) were applied for statistical work-up.

Results: All three substances significantly reduced the number of histologically visible inflammatory cells compared to the control group (p<0.05).

Conclusions: In the present study, topical allopurinol was as effective as established drugs, namely steroids and acetylcysteine, in the early treatment of experimental alkali corneal burns.

MeSH terms

  • Acetylcysteine / administration & dosage*
  • Acetylcysteine / therapeutic use
  • Administration, Topical
  • Alkalies*
  • Allopurinol / administration & dosage*
  • Allopurinol / therapeutic use
  • Animals
  • Anti-Inflammatory Agents / administration & dosage*
  • Anti-Inflammatory Agents / therapeutic use
  • Burns, Chemical / drug therapy*
  • Burns, Chemical / pathology
  • Drug Therapy, Combination
  • Enzyme Inhibitors / administration & dosage*
  • Enzyme Inhibitors / therapeutic use
  • Eye Burns / chemically induced*
  • Eye Burns / drug therapy*
  • Eye Burns / pathology
  • Free Radical Scavengers / administration & dosage*
  • Free Radical Scavengers / therapeutic use
  • Male
  • Ophthalmic Solutions
  • Pilot Projects
  • Prednisolone / administration & dosage*
  • Prednisolone / analogs & derivatives*
  • Prednisolone / therapeutic use
  • Rats
  • Rats, Wistar
  • Treatment Outcome

Substances

  • Alkalies
  • Anti-Inflammatory Agents
  • Enzyme Inhibitors
  • Free Radical Scavengers
  • Ophthalmic Solutions
  • Allopurinol
  • prednisolone acetate
  • Prednisolone
  • Acetylcysteine