Upregulation of the oncogene c-myc in Barrett's adenocarcinoma: induction of c-myc by acidified bile acid in vitro

Gut. 2003 Feb;52(2):174-80. doi: 10.1136/gut.52.2.174.

Abstract

Background and aims: C-myc over expression is implicated in malignancy although to date this has not been studied in Barrett's metaplasia. We sought to determine c-myc expression in the malignant progression of Barrett's metaplasia and whether it may be induced by bile acids seen in gastro-oesophageal refluxate.

Methods: C-myc protein and mRNA levels were assessed in 20 Barrett's metaplasia and 20 oesophageal adenocarcinoma samples by western blotting and real time polymerase chain reaction. Levels of c-myc and proliferation were also assessed in cell lines OE21, OE33, SW-480, and TE-7 stimulated with pulses or continuous exposure to the bile acids deoxycholic acid and chenodeoxycholic acid.

Results: C-myc protein was upregulated in 50% of Barrett's metaplasia and 90% of oesophageal adenocarcinoma samples compared with squamous, gastric, and duodenal controls. C-myc immunolocalisation in Barrett's metaplasia revealed discrete nuclear localisation, becoming more diffuse with progression from low to high grade dysplasia to adenocarcinoma. Both continual and pulsed bile acid induced c-myc at pH 4, with no effect at pH 7 or with acidified media alone. Pulsed bile acid treatment induced proliferation (p<0.05); in contrast, continuous exposure led to suppression of proliferation (p<0.05).

Conclusions: We have shown upregulation of c-myc with malignant progression of Barrett's metaplasia and suggest that acidified bile may be a novel agent responsible for induction of this oncogene.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenocarcinoma / genetics*
  • Adenocarcinoma / pathology
  • Barrett Esophagus / genetics*
  • Barrett Esophagus / pathology
  • Bile Acids and Salts / pharmacology*
  • Blotting, Western / methods
  • Cell Division
  • Chenodeoxycholic Acid / pharmacology
  • Deoxycholic Acid / pharmacology
  • Esophageal Neoplasms / genetics*
  • Esophageal Neoplasms / pathology
  • Fluorescent Antibody Technique / methods
  • Gastroesophageal Reflux / metabolism
  • Gene Expression Regulation / drug effects
  • Genes, myc / drug effects
  • Genes, myc / genetics*
  • Humans
  • Immunohistochemistry / methods
  • Polymerase Chain Reaction / methods
  • Tumor Cells, Cultured
  • Up-Regulation / drug effects*
  • Up-Regulation / genetics

Substances

  • Bile Acids and Salts
  • Deoxycholic Acid
  • Chenodeoxycholic Acid