Transcriptional activation by AP-2alpha is modulated by the oncogene DEK

Nucleic Acids Res. 2003 Mar 1;31(5):1571-5. doi: 10.1093/nar/gkg247.

Abstract

Cell differentiation and development are highly regulated processes at the transcriptional level. One of the main transcription factors that regulate these processes is AP-2alpha, a cell-type specific protein required for vertebrate development and embryogenesis. AP-2alpha also regulates apoptosis and cell-cycle specific events by interacting with the oncogene c-Myc. In searching for novel AP-2alpha- interacting factors, using an affinity chromatography approach, we have observed that oncoprotein DEK interacts with AP-2alpha in vitro. The existence of an interaction between AP-2alpha and DEK in cellular cultures was demonstrated by expression of a tagged AP-2alpha form followed by immunodetection. By transient co-expression experiments using a reporter for APOE promoter activity we have found that DEK stimulates the transactivation activity of AP-2alpha over APOE promoter. Finally, electrophoretic mobility shift assays suggested that DEK enhances the DNA-binding activity of AP-2alpha. Our data suggest a novel cellular function of DEK as a transcriptional co-activator.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apolipoproteins E / genetics
  • Chromatography, Affinity
  • Chromosomal Proteins, Non-Histone*
  • DNA / metabolism
  • DNA-Binding Proteins / genetics
  • DNA-Binding Proteins / metabolism*
  • Electrophoretic Mobility Shift Assay
  • Humans
  • Oncogene Proteins / genetics
  • Oncogene Proteins / metabolism*
  • Oncogene Proteins / pharmacology
  • Poly-ADP-Ribose Binding Proteins
  • Promoter Regions, Genetic / genetics
  • Protein Binding / drug effects
  • Recombinant Fusion Proteins / genetics
  • Recombinant Fusion Proteins / metabolism
  • Recombinant Fusion Proteins / pharmacology
  • Transcription Factor AP-2
  • Transcription Factors / genetics
  • Transcription Factors / metabolism*
  • Transcriptional Activation
  • Transfection
  • Tumor Cells, Cultured

Substances

  • Apolipoproteins E
  • Chromosomal Proteins, Non-Histone
  • DNA-Binding Proteins
  • DEK protein, human
  • Oncogene Proteins
  • Poly-ADP-Ribose Binding Proteins
  • Recombinant Fusion Proteins
  • TFAP2A protein, human
  • Transcription Factor AP-2
  • Transcription Factors
  • DNA