Synthesis and in vitro leishmanicidal activity of some hydrazides and their analogues

Bioorg Med Chem. 2003 Apr 3;11(7):1381-7. doi: 10.1016/s0968-0896(02)00611-9.

Abstract

Twenty-one hydrazides were synthesized by treating different esters with hydrazine hydrate. Substituted hydrazides were obtained by treating hydrazides with alkyl/aryl/acyl halides. Some of these compounds exhibit potential in vitro leishmanicidal activity. The structures of all the synthesized compounds were confirmed by spectroscopic analysis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alkylation
  • Animals
  • Antiprotozoal Agents / chemical synthesis*
  • Antiprotozoal Agents / pharmacology*
  • Hydrazines / chemical synthesis*
  • Hydrazines / pharmacology*
  • Indicators and Reagents
  • Leishmania major / drug effects*
  • Magnetic Resonance Spectroscopy
  • Solvents

Substances

  • Antiprotozoal Agents
  • Hydrazines
  • Indicators and Reagents
  • Solvents
  • hydrazine