Single-chain Fv multimers of the anti-neuraminidase antibody NC10: the residue at position 15 in the V(L) domain of the scFv-0 (V(L)-V(H)) molecule is primarily responsible for formation of a tetramer-trimer equilibrium

Protein Eng. 2003 Jan;16(1):47-56. doi: 10.1093/proeng/gzg006.

Abstract

Single-chain variable fragment of the murine monoclonal antibody NC10 specific to influenza virus N9 neuraminidase, joined directly in the V(L) to V(H) orientation (scFv-0), forms an equilibrium mixture of tetramer and trimer with the tetramer as the preferred multimeric species. In contrast, the V(H)-V(L) isomer was previously shown to exist exclusively as a trimer. Computer-generated trimeric and tetrameric scFv models, based on the refined crystal structure for NC10 Fv domain, were constructed and used to evaluate factors influencing the transition between V(L)-V(H) trimer and tetramer. These model structures indicated that steric restrictions between loops spanning amino acid residues L55-L59 and L13-L17 from the two adjacent V(L) domains within the V(L)-V(H) trimer were responsible for four scFv-0 molecules assembling to form a tetramer. In particular, leucine at position L15 and glutamate at position L57 appeared to interfere significantly with each other. To minimize this steric interference, the site-directed mutagenesis technique was used to construct several NC10 scFv-0 clones with mutations at these positions. Size-exclusion chromatographic analyses revealed that several of these mutations resulted in the production of NC10 scFv-0 proteins with significantly altered tetramer-trimer equilibrium ratios. In particular, introduction of a polar residue, such as asparagine or threonine, at position L15 generated a highly stable NC10 scFv-0 trimer.

MeSH terms

  • Amino Acid Sequence
  • Amino Acid Substitution
  • Animals
  • Antibodies / chemistry*
  • Antibodies / genetics
  • Antibodies / metabolism
  • Chromatography, Gel
  • Electrophoresis, Polyacrylamide Gel
  • Glutamic Acid / chemistry
  • Glutamic Acid / genetics
  • Immunoglobulin Variable Region / chemistry*
  • Immunoglobulin Variable Region / metabolism
  • Kinetics
  • Leucine / chemistry
  • Leucine / genetics
  • Mice
  • Models, Molecular
  • Mutagenesis, Site-Directed
  • Neuraminidase / immunology*
  • Protein Binding
  • Protein Conformation
  • Protein Structure, Tertiary
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / genetics
  • Recombinant Proteins / metabolism

Substances

  • Antibodies
  • Immunoglobulin Variable Region
  • Recombinant Proteins
  • Glutamic Acid
  • Neuraminidase
  • Leucine