No effect of an L-arginine-enriched medical food (HeartBars) on endothelial function and platelet aggregation in subjects with hypercholesterolemia

Am Heart J. 2003 Mar;145(3):E15. doi: 10.1067/mhj.2003.160.

Abstract

Background: Providing L-arginine as a precursor for nitric oxide has been proposed to improve endothelial function in populations at high risk for cardiovascular events. We studied the effects of dietary L-arginine supplementation with HeartBars (a medical food rich in L-arginine, Cooke Pharma, Belmont, Calif) on flow-mediated dilation and markers of endothelial function in subjects with hypercholesterolemia.

Methods: We randomly assigned 47 subjects with hypercholesterolemia to receive one HeartBar containing 3.3 g L-arginine each, or a placebo bar, consumed twice daily for 2 weeks. Flow-mediated dilation, platelet aggregation studies, and soluble levels of endothelial and platelet adhesion molecules were obtained before and after the 2-week treatment period.

Results: Baseline and follow-up levels of L-arginine were 78.5 +/- 28.2 micromol/L and 80.7 +/- 26.7 micromol/L, respectively (P =.54). The HeartBar group had no improvement in flow-mediated dilation; changes in brachial artery diameter at baseline and follow-up were 5.52% +/- 3.32% and 4.96% +/- 2.39%, respectively. There were also no changes in the soluble levels of E-selectin and P-selectin by treatment group.

Conclusions: In our study, 2 weeks of HeartBar supplementation in subjects with hypercholesterolemia showed no favorable effects on endothelial or platelet function.

Publication types

  • Clinical Trial
  • Comparative Study
  • Multicenter Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Ambulatory Care
  • Arginine / metabolism
  • Arginine / pharmacology
  • Arginine / therapeutic use*
  • Brachial Artery / drug effects
  • Brachial Artery / physiology
  • Endothelium, Vascular / drug effects*
  • Endothelium, Vascular / physiology
  • Female
  • Food, Fortified*
  • Humans
  • Hypercholesterolemia / diet therapy*
  • Male
  • Middle Aged
  • Nitric Oxide / biosynthesis
  • Nitric Oxide / therapeutic use
  • Platelet Aggregation / drug effects*
  • Platelet Aggregation / physiology
  • Prodrugs / metabolism
  • Prodrugs / pharmacology
  • Prodrugs / therapeutic use
  • Regional Blood Flow / drug effects
  • Regional Blood Flow / physiology
  • Treatment Outcome
  • Vasodilation / drug effects
  • Vasodilation / physiology

Substances

  • Prodrugs
  • Nitric Oxide
  • Arginine