A simplified model of the binding interaction between stromal cell-derived factor-1 chemokine and CXC chemokine receptor 4

Protein Pept Lett. 2003 Apr;10(2):133-8. doi: 10.2174/0929866033479022.

Abstract

We have synthesised the CXC chemokine receptor 4 (29-39) peptide, CXCR4[29-39]. This peptide is located in the N-terminal region of the receptor and is likely to be involved in the docking step of the receptor interaction with its natural ligand stromal cell-derived factor-1 chemokine, SDF-1. Preliminary experiments, performed in the presence of micellar detergents to model a membrane-like environment, show that the (1-17) segment of SDF-1 binds to CXCR4[29-39].

MeSH terms

  • Animals
  • Chemokine CXCL12
  • Chemokines, CXC / metabolism*
  • Fluorescence
  • Humans
  • Phenylalanine / metabolism
  • Receptors, CXCR4 / metabolism*

Substances

  • CXCL12 protein, human
  • Chemokine CXCL12
  • Chemokines, CXC
  • Receptors, CXCR4
  • Phenylalanine