Dose-dependent severe cutaneous reactions to imatinib

Br J Cancer. 2003 Apr 22;88(8):1157-9. doi: 10.1038/sj.bjc.6600893.

Abstract

The protein kinase inhibitor imatinib has been approved as an efficient anticancer drug with common but mild cutaneous toxicities. We here report on two out of four melanoma patients treated with high-dose imatinib presenting with severe and strongly dose-dependent skin eruptions, suggesting a cutaneous reactivity pattern different from allergic hypersensitivity.

Publication types

  • Case Reports

MeSH terms

  • Adult
  • Aged
  • Antineoplastic Agents / toxicity*
  • Benzamides
  • Drug Hypersensitivity* / pathology*
  • Female
  • Humans
  • Imatinib Mesylate
  • Male
  • Middle Aged
  • Piperazines / toxicity*
  • Pyrimidines / toxicity*
  • Skin Diseases / chemically induced*
  • Skin Diseases / pathology

Substances

  • Antineoplastic Agents
  • Benzamides
  • Piperazines
  • Pyrimidines
  • Imatinib Mesylate