Inhibition of p53-induced apoptosis without affecting expression of p53-regulated genes

Proc Natl Acad Sci U S A. 2003 May 27;100(11):6718-23. doi: 10.1073/pnas.1031695100. Epub 2003 May 12.

Abstract

Using DNA microarray and clustering of expressed genes we have analyzed the mechanism of inhibition of wild-type p53-induced apoptosis by the cytokine interleukin 6 (IL-6) and the calcium mobilizer thapsigargin (TG). Clustering analysis of 1,786 genes, the expression level of which changed after activation of wild-type p53 in the absence or presence of IL-6 or TG, showed that these compounds did not cause a general inhibition of the ability of p53 to up-regulate or down-regulate gene expression. Expression of various p53 targets implicated as mediators of p53-induced apoptosis was also not affected by IL-6 or TG. These compounds thus can bypass the effect of wild-type p53 on gene expression and inhibit apoptosis. IL-6 and TG activated different p53-independent pathways of gene expression that include up-regulation of antiapoptotic genes. IL-6 and TG also activated different differentiation-associated genes. The ability of compounds such as cytokines and calcium mobilizers to inhibit p53-mediated apoptosis without generally inhibiting gene expression regulated by p53 can facilitate tumor development and tumor resistance to radiation and chemotherapy in cells that retain wild-type p53.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Apoptosis / physiology*
  • Base Sequence
  • Blotting, Western
  • Cell Differentiation
  • Cluster Analysis
  • DNA Primers
  • Gene Expression Regulation / drug effects
  • Gene Expression Regulation / physiology*
  • Interleukin-6 / physiology
  • Molecular Sequence Data
  • Oligonucleotide Array Sequence Analysis
  • Reverse Transcriptase Polymerase Chain Reaction
  • Thapsigargin / pharmacology
  • Tumor Cells, Cultured
  • Tumor Suppressor Protein p53 / physiology*

Substances

  • DNA Primers
  • Interleukin-6
  • Tumor Suppressor Protein p53
  • Thapsigargin

Associated data

  • GENBANK/AF067774
  • RefSeq/NM_009735