(Patho)physiological implications of the novel epithelial Ca2+ channels TRPV5 and TRPV6

Pflugers Arch. 2003 Jul;446(4):401-9. doi: 10.1007/s00424-003-1038-7. Epub 2003 May 13.

Abstract

The epithelial Ca(2+) channels TRPV5 and TRPV6 constitute the apical Ca(2+) entry mechanism in active Ca(2+) (re)absorption. These two members of the superfamily of transient receptor potential (TRP) channels were cloned from the vitamin-D-responsive epithelia of kidney and small intestine and subsequently identified in other tissues such as bone, pancreas and prostate. These channels are regulated by vitamin D as exemplified in animal models of vitamin-D-deficiency rickets. In addition, the epithelial Ca(2+) channels might be involved in the multifactorial pathogenesis of disorders ranging from idiopathic hypercalciuria, stone disease and postmenopausal osteoporosis. This review highlights the emerging (patho)physiological implications of these epithelial Ca(2+) channels.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Calcium / metabolism*
  • Calcium Channels / physiology*
  • Epithelial Cells / physiology*
  • Humans
  • Metabolic Diseases / metabolism
  • Metabolic Diseases / physiopathology*
  • TRPV Cation Channels

Substances

  • Calcium Channels
  • TRPV Cation Channels
  • TRPV5 protein, human
  • TRPV6 channel
  • Calcium