Decreased lymphocyte 3H-paroxetine binding in obsessive-compulsive disorder

Neuropsychobiology. 2003;47(3):128-30. doi: 10.1159/000070580.

Abstract

The pathophysiology of obsessive-compulsive disorder (OCD) is mainly focused on the serotonin (5-HT) system and transporter. The presence of this structure in blood lymphocytes prompted us to investigate it, by means of the specific binding of (3)H-paroxetine ((3)H-PAR), in a group of drug-free OCD patients as compared with healthy control subjects matched for sex and age. Lymphocyte membranes and (3)H-PAR binding were carried out according to standard protocols. The results showed that the patients had a statistically significant lower density of (3)H-PAR-binding sites than the control subjects. On one hand, this finding confirms previous data of an abnormal platelet 5-HT transporter in OCD, on the other it provides the possibility to explore the regulation of this structure in this and other disorders, since lymphocytes are nucleate cells.

MeSH terms

  • Adult
  • Antidepressive Agents, Second-Generation / pharmacokinetics*
  • Antidepressive Agents, Second-Generation / therapeutic use
  • Binding Sites
  • Carrier Proteins / metabolism
  • Carrier Proteins / physiology*
  • Female
  • Humans
  • Lymphocytes / metabolism*
  • Male
  • Membrane Glycoproteins / metabolism
  • Membrane Glycoproteins / physiology*
  • Membrane Transport Proteins*
  • Nerve Tissue Proteins*
  • Obsessive-Compulsive Disorder / drug therapy
  • Obsessive-Compulsive Disorder / metabolism*
  • Obsessive-Compulsive Disorder / physiopathology*
  • Paroxetine / pharmacokinetics*
  • Paroxetine / therapeutic use
  • Serotonin Plasma Membrane Transport Proteins

Substances

  • Antidepressive Agents, Second-Generation
  • Carrier Proteins
  • Membrane Glycoproteins
  • Membrane Transport Proteins
  • Nerve Tissue Proteins
  • SLC6A4 protein, human
  • Serotonin Plasma Membrane Transport Proteins
  • Paroxetine