Increased expression of cyclin E is associated with an increased resistance to doxorubicin in rat fibroblasts

Br J Cancer. 2003 Jun 16;88(12):1956-62. doi: 10.1038/sj.bjc.6600970.

Abstract

Cell cycle progression in eukaryotic cells is regulated by a family of cyclin-dependent kinases (CDKs). Cyclin E is a regulatory subunit of CDK2 and drives cells from G1 to S phase. Increased expression of cyclin E is a frequent event in human malignancies and has been associated with poor prognosis in various cancers. In this study, we evaluated the effects of cyclin E-overexpression on the sensitivity of rat fibroblasts to anticancer drugs. Cyclin E-overexpressing cells were less sensitive to doxorubicin-induced inhibition of cell growth but not to other antineoplastic drugs, such as paclitaxel, vincristine, etoposide and methotrexate. Cyclin E-overexpressing fibroblasts also displayed a reduction in ROS levels and a significantly lower increase following doxorubicin treatment compared with vector control cells. The expression of manganese superoxide dismutase (MnSOD) and its activity were increased (about 1.3-fold) in cyclin E-overexpressing derivatives compared with control cells. These results suggest that cyclin E overexpression might reduce tumour cells sensitivity to doxorubicin by affecting the expression of MnSOD and that determination of cyclin E expression levels might help to select patients to be treated with an anthracycline-based antineoplastic therapy.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antineoplastic Agents / pharmacology*
  • Cell Division
  • Cells, Cultured
  • Cyclin E / biosynthesis*
  • Doxorubicin / pharmacology*
  • Drug Resistance*
  • Fibroblasts / drug effects*
  • Fibroblasts / metabolism*
  • Rats
  • Reactive Oxygen Species / metabolism
  • Superoxide Dismutase / biosynthesis

Substances

  • Antineoplastic Agents
  • Cyclin E
  • Reactive Oxygen Species
  • Doxorubicin
  • Superoxide Dismutase