The alpha-L-ribo-isomers of RNA and LNA (locked nucleic acid)

Nucleic Acids Res Suppl. 2001:(1):25-6. doi: 10.1093/nass/1.1.25.

Abstract

The phosphoramidite approach has been used for the automated synthesis of alpha-L-LNA, alpha-L-RNA, and oligomers composed of mixtures of alpha-L-LNA, alpha-L-RNA and DNA monomers. Binding studies revealed very efficient recognition of single-stranded DNA and RNA target oligonucleotide strands. alpha-L-LNAs were shown to be significantly stabilized towards 3'-exonucleolytic degradation. Duplexes formed between RNA and alpha-L-LNA induced E. coli RNase H-mediated RNA cleavage, albeit very slow, at high enzyme concentration.

MeSH terms

  • DNA / chemistry
  • Endoribonucleases / metabolism
  • Escherichia coli / enzymology
  • Exonucleases / metabolism
  • Nucleic Acid Hybridization
  • Nucleic Acids / chemistry*
  • Nucleic Acids / metabolism
  • RNA / chemistry*
  • RNA / metabolism
  • Stereoisomerism

Substances

  • Nucleic Acids
  • RNA
  • DNA
  • Endoribonucleases
  • Exonucleases