P-locus is a target for the melanogenic effects of MC-1R signaling: a possible control point for facultative pigmentation

Ann N Y Acad Sci. 2003 Jun:994:373-7. doi: 10.1111/j.1749-6632.2003.tb03202.x.

Abstract

Melanocortin receptor type 1 (MC-1R) is an important control point for ultraviolet ray (UVR)-induced tanning response in the skin. In this study, we show that p-locus is a downstream target for MC-1R signaling. The expression of p-locus was up-regulated by alpha-MSH as well as db-cAMP, a synthetic analogue of cAMP that mimics activation of MC-1R. Furthermore, p-locus transcript abundance was significantly increased in epidermal melanocytes of white skin with facultative (UVR-induced) pigmentation. Because p-locus product is essential for pigmentation and also has been shown to be highly polymorphic in human population, we propose that the pigmentary response to the melanocortin peptides/UVR would be affected not only by MC-1R mutations but also by the functionality of p-locus product. These factors together could account for the many different levels of tanning ability seen in the white population.

Publication types

  • Review

MeSH terms

  • Bucladesine / metabolism
  • Gene Expression Regulation*
  • Humans
  • Receptors, Corticotropin / genetics
  • Receptors, Corticotropin / metabolism*
  • Receptors, Melanocortin
  • Signal Transduction / physiology*
  • Skin / cytology
  • Skin / metabolism
  • Skin / radiation effects
  • Skin Pigmentation / physiology*
  • Ultraviolet Rays
  • alpha-MSH / metabolism*

Substances

  • Receptors, Corticotropin
  • Receptors, Melanocortin
  • alpha-MSH
  • Bucladesine