Alpha-galactosylceramide (KRN7000) suppression of chemical- and oncogene-dependent carcinogenesis

Proc Natl Acad Sci U S A. 2003 Aug 5;100(16):9464-9. doi: 10.1073/pnas.1630663100. Epub 2003 Jul 16.

Abstract

Recent studies have revealed significant efficacy of the marine sponge glycolipid, alpha-galactosylceramide (alpha-GalCer), in treatment of experimental metastatic cancers, infections, and autoimmune diseases. However, the capacity of alpha-GalCer to prevent tumor development had never, to our knowledge, been evaluated in mouse models of chemical- and oncogene-dependent carcinogenesis. In this study, we demonstrate that long-term administration of soluble alpha-GalCer, spanning the time of tumor initiation, inhibits primary tumor formation in three different models: methylcholanthrene-induced sarcomas, mammary carcinomas in Her-2/neu transgenic mice, and spontaneous sarcomas in p53-/- mice. Weekly treatment of mice with alpha-GalCer maintained lymphoid tissue natural killer cell and T cell activation and elevated serum IFN-gamma and IL-4 concentrations. Consistent with the antimetastatic activity of alpha-GalCer, prevention of methylcholanthrene-induced sarcoma was IFN-gammaand tumor necrosis factor-related apoptosis-inducing ligand dependent, but not perforin-dependent. Taken together, our results demonstrate that NK1.1+alphabetaTCR+ cell-based immune therapy can inhibit primary tumorigenesis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antineoplastic Agents / pharmacology*
  • Apoptosis
  • Dose-Response Relationship, Drug
  • Enzyme-Linked Immunosorbent Assay
  • Fibrosarcoma / metabolism
  • Flow Cytometry
  • Galactosylceramides / pharmacology*
  • Genes, p53
  • Humans
  • Interferon-gamma / genetics
  • Interleukin-12 / metabolism
  • Interleukin-4 / metabolism
  • Ligands
  • Methylcholanthrene / pharmacology
  • Mice
  • Mice, Inbred BALB C
  • Mice, Inbred C57BL
  • Mice, Transgenic
  • Mutation
  • Neoplasms / chemically induced*
  • Neoplasms / genetics
  • Neoplasms / prevention & control*
  • Receptor, ErbB-2 / genetics
  • Time Factors
  • Tumor Cells, Cultured
  • Tumor Suppressor Protein p53 / genetics

Substances

  • Antineoplastic Agents
  • Galactosylceramides
  • Ligands
  • Tumor Suppressor Protein p53
  • Interleukin-12
  • Interleukin-4
  • Methylcholanthrene
  • Interferon-gamma
  • Receptor, ErbB-2
  • KRN 7000