The immune response modifier and Toll-like receptor 7 agonist S-27609 selectively induces IL-12 and TNF-alpha production in CD11c+CD11b+CD8- dendritic cells

J Immunol. 2003 Aug 1;171(3):1156-63. doi: 10.4049/jimmunol.171.3.1156.

Abstract

IL-12 and TNF-alpha production by dendritic cells (DCs) is a critical step in the initiation of local inflammation and adaptive immune responses. We show in this study that a small molecule immune response modifier that is a Toll-like receptor 7 (TLR7) agonist induces IL-12 and TNF-alpha production from murine CD11c(+)CD11b(+)CD8(-) DCs, a subset not previously known for this activity. Stimulation of these DCs through TLR7 in vivo induces significant cytokine production even 12 h after initial stimulation, as well as migration of the DC into T cell zones of the lymphoid tissue. In contrast, stimulation through TLR4 and TLR9 induced IL-12 production predominantly from CD8(+) DCs, consistent with previously published data. All TLR stimuli induced the increase in surface expression of the activation markers B7-1, B7-2, and class II in both CD8(+) and CD8(-) DCs, demonstrating that CD8(+) DCs do respond to TLR7-mediated stimuli. To date this is the only known stimuli to induce preferential cytokine production from CD8(-) DCs. Given the efficacy of TLR7 agonists as antiviral agents, the data collectively indicate that stimulation of CD8(-) DCs through TLR7 most likely plays a role in the generation of antiviral immune responses.

MeSH terms

  • Aminoquinolines / administration & dosage*
  • Animals
  • CD11b Antigen / biosynthesis*
  • CD11c Antigen / biosynthesis*
  • CD8 Antigens / biosynthesis
  • Cell Line
  • Cell Movement / immunology
  • Cytokines / biosynthesis
  • DNA-Binding Proteins / agonists
  • DNA-Binding Proteins / physiology
  • Dendritic Cells / drug effects
  • Dendritic Cells / immunology*
  • Dendritic Cells / metabolism
  • Female
  • Humans
  • Immunologic Factors / pharmacology*
  • Injections, Intravenous
  • Interleukin-12 / biosynthesis*
  • Membrane Glycoproteins / agonists*
  • Membrane Glycoproteins / physiology
  • Mice
  • Mice, Inbred C57BL
  • Myeloid Cells / drug effects
  • Myeloid Cells / immunology
  • Myeloid Cells / metabolism
  • Receptors, Cell Surface / agonists*
  • Receptors, Cell Surface / physiology
  • Spleen / cytology
  • Spleen / drug effects
  • Spleen / immunology
  • Spleen / metabolism
  • T-Lymphocyte Subsets / drug effects
  • T-Lymphocyte Subsets / immunology
  • Toll-Like Receptor 7
  • Toll-Like Receptor 9
  • Tumor Necrosis Factor-alpha / biosynthesis*

Substances

  • 4-amino-alpha,alpha,2-trimethyl-1H-imidazo(4,5-c)quinoline-1-ethanol
  • Aminoquinolines
  • CD11b Antigen
  • CD11c Antigen
  • CD8 Antigens
  • Cytokines
  • DNA-Binding Proteins
  • Immunologic Factors
  • Membrane Glycoproteins
  • Receptors, Cell Surface
  • TLR9 protein, human
  • Tlr7 protein, mouse
  • Tlr9 protein, mouse
  • Toll-Like Receptor 7
  • Toll-Like Receptor 9
  • Tumor Necrosis Factor-alpha
  • Interleukin-12