Single-dose pharmacokinetics of ofloxacin during continuous venovenous hemofiltration in critical care patients

Am J Kidney Dis. 2003 Aug;42(2):310-4. doi: 10.1016/s0272-6386(03)00656-5.

Abstract

Background: Ofloxacin is a quinolone administered to patients with severe infections. Pharmacokinetic data on ofloxacin in critically ill patients on renal replacement therapy are sparse and conflicting.

Methods: Eight patients with anuric acute renal failure were administered 400 mg of ofloxacin intravenously. The pharmacokinetics of ofloxacin was analyzed during continuous venovenous hemofiltration (CVVH) with a high-flux polysulfone membrane. Serum and ultrafiltrate levels of ofloxacin were measured by means of high-performance liquid chromatography.

Results: Mean serum ofloxacin concentration peak was 5.5 +/- 0.7 mg/L. Elimination half-life, hemofiltration clearance, and total removal were 2.8 +/- 0.5 hours, 89.9 +/- 4.5 mL/min, and 76.9% +/- 7.1%, respectively.

Conclusion: Ofloxacin is significantly and rapidly eliminated by CVVH with a high-flux polysulfone membrane.

MeSH terms

  • Acute Kidney Injury / complications
  • Acute Kidney Injury / drug therapy*
  • Adult
  • Aged
  • Anti-Infective Agents / pharmacokinetics*
  • Anti-Infective Agents / therapeutic use
  • Chromatography, High Pressure Liquid
  • Critical Care*
  • Female
  • Gram-Negative Bacterial Infections / complications
  • Gram-Negative Bacterial Infections / drug therapy*
  • Half-Life
  • Hemofiltration*
  • Humans
  • Male
  • Metabolic Clearance Rate
  • Middle Aged
  • Ofloxacin / pharmacokinetics*
  • Ofloxacin / therapeutic use

Substances

  • Anti-Infective Agents
  • Ofloxacin