Flufenacet herbicide treatment phenocopies the fiddlehead mutant in Arabidopsis thaliana

Pest Manag Sci. 2003 Aug;59(8):847-56. doi: 10.1002/ps.714.

Abstract

In order to study the mode of action of herbicides we conducted a pilot study analysing phenotype and gene expression of flufenacet- and benfuresate-treated Arabidopsis thaliana (L) Heynhoe plants. Treatments with either herbicide caused phenocopies of the known Arabidopsis mutant fiddlehead, displaying fused organs and the typical fiddlehead-like inflorescence. Herbicide treatments of other plant species, including monocots, also gave rise to analogous organ fusions, indicating the presence of the target in a broad range of plants. Furthermore, many other herbicides with a proposed similar mode of action, eg chloroacetanilides, produced comparable fusion phenotypes in plants. The fiddlehead gene encodes a putative very-long-chain fatty acid elongase (VLCFAE), which corroborates earlier biochemical results pointing to the inhibition of VLCFA synthesis as mode of action of flufenacet. Gene expression profiles of herbicide-treated plants using the first 8247 gene Arabidopsis gene array of Affymetrix provided additional clues in support of inhibition of VLCFA synthesis. We discuss fiddlehead-like elongases as plant specific targets for flufenacet and many other herbicides.

MeSH terms

  • Acetamides / chemistry
  • Acetamides / pharmacology*
  • Amino Acid Sequence
  • Arabidopsis / drug effects*
  • Arabidopsis / enzymology
  • Arabidopsis / genetics*
  • Arabidopsis Proteins / genetics*
  • Benzofurans / chemistry
  • Benzofurans / pharmacology*
  • Gene Expression Profiling
  • Gene Expression Regulation, Plant / drug effects*
  • Herbicides / chemistry
  • Herbicides / pharmacology*
  • Molecular Sequence Data
  • Molecular Structure
  • Oligonucleotide Array Sequence Analysis
  • Phenotype
  • Phylogeny
  • Sulfonic Acids / chemistry
  • Sulfonic Acids / pharmacology*
  • Thiadiazoles / chemistry
  • Thiadiazoles / pharmacology*

Substances

  • Acetamides
  • Arabidopsis Proteins
  • At2g26250 protein, Arabidopsis
  • Benzofurans
  • Herbicides
  • Sulfonic Acids
  • Thiadiazoles
  • FOE 5043
  • benfuresate