p73 is regulated by phosphorylation at the G2/M transition

J Biol Chem. 2003 Dec 5;278(49):49196-202. doi: 10.1074/jbc.M304921200. Epub 2003 Aug 13.

Abstract

p73 is a p53 paralog that encodes proapoptotic (transactivation-competent (TA)) and antiapoptotic (dominant negative) isoforms. TAp73 transcription factors mediate cell cycle arrest and/or apoptosis in response to DNA damage and are involved in developmental processes in the central nervous system and the immune system. p73 proteins may also play a role in the regulation of cell growth. Indeed, p73 expression is itself modulated during the cell cycle and TAp73 proteins accumulate in S phase cells. In addition, the function of p73 proteins is also regulated by post-translational modifications and protein-protein interactions in different cellular and pathophysiological contexts. Here we show that p73 is a physiological target of the p34cdc2-cyclin B mitotic kinase complex in vivo. Both p73beta and p73alpha isoforms are hyperphosphorylated in normal mitotic cells and during mitotic arrest induced by microtubule-targeting drugs. p34cdc2-cyclin B phosphorylates and associates with p73 in vivo, which results in a decreased ability of p73 to both bind DNA and activate transcription in mitotic cells. Indeed, p73 is excluded from condensed chromosomes in meta- and anaphase, redistributes throughout the mitotic cytoplasm, and unlike p53, shows no association with centrosomes. Together these results indicate that M phase-specific phosphorylation of p73 by p34cdc2-cyclin B is associated with negative regulation of its transcriptional activating function.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Line, Tumor
  • Cyclin B / metabolism
  • Cyclin-Dependent Kinase 4
  • Cyclin-Dependent Kinases / metabolism
  • DNA-Binding Proteins / physiology*
  • G2 Phase*
  • Genes, Tumor Suppressor
  • Humans
  • Mitosis*
  • Nuclear Proteins / physiology*
  • Phosphorylation
  • Proto-Oncogene Proteins*
  • Tumor Protein p73
  • Tumor Suppressor Proteins

Substances

  • Cyclin B
  • DNA-Binding Proteins
  • Nuclear Proteins
  • Proto-Oncogene Proteins
  • TP73 protein, human
  • Tumor Protein p73
  • Tumor Suppressor Proteins
  • CDK4 protein, human
  • Cyclin-Dependent Kinase 4
  • Cyclin-Dependent Kinases

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