Vigabatrin does not affect the intestinal absorption of phenytoin in rat duodeno-jejunal loops in situ

Pharmacol Res. 1992 Sep;26(2):201-5. doi: 10.1016/s1043-6618(05)80133-1.

Abstract

The antiepileptic drug vigabatrin (GVG) is known to decrease significantly the serum concentration of concurrently administered phenytoin (PHT) in epileptic patients. To assess a possible mechanism for this interaction, the effect of GVG on the intestinal absorption of PHT was investigated by means of circulation experiments in an in situ rat duodeno-jejunal loop. GVG did not affect the rate of disappearance of PHT from the loop perfusing medium, providing evidence against occurrence of GVG-induced impairment of PHT absorption.

MeSH terms

  • Aminocaproates / pharmacology*
  • Animals
  • Anticonvulsants / pharmacology*
  • Duodenum / metabolism
  • Intestinal Absorption / drug effects*
  • Jejunum / metabolism
  • Male
  • Phenytoin / metabolism*
  • Rats
  • Rats, Sprague-Dawley
  • Vigabatrin

Substances

  • Aminocaproates
  • Anticonvulsants
  • Phenytoin
  • Vigabatrin