Effects of L-threo- and erythro-3,4-dihydroxyphenylserine on learning performance and concentrations of brain noradrenaline and its metabolites in rats

Pharmacol Biochem Behav. 1992 Sep;43(1):215-21. doi: 10.1016/0091-3057(92)90660-8.

Abstract

Effects of L-threo and L-erythro-3,4-dihydroxyphenylserine [DOPS, precursor amino acids for noradrenaline (NA)] on the learning performance in a maze paradigm designed to model on the water maze paradigm using a multicomputerized behavioral analysis system were studied. A marked facilitation of learning performance was observed in rats after an intraventricular injection of 5 micrograms L-threo-DOPS (the s-NA precursor), and this effect was inhibited by a simultaneous administration of 1 or 2 micrograms propranolol (a beta-adrenergic antagonist). As concentrations of brain NA, 3-methoxy-4-hydroxyphenylglycol, and normethanephrine were increased by the injection of 5 micrograms L-threo-DOPS, the effect seemed to be derived from activation of beta-adrenoceptors in the CNS by the formed s-NA. On the other hand, an intraventricular injection of 5 micrograms L-erythro-DOPS (the r-NA precursor) attenuated the learning performance, and this effect was probably caused by the formed r-NA from L-erythro-DOPS.

MeSH terms

  • Animals
  • Biogenic Monoamines / metabolism
  • Brain Chemistry / drug effects*
  • Droxidopa / pharmacology*
  • Injections, Intraventricular
  • Learning / drug effects*
  • Male
  • Motor Activity / drug effects
  • Norepinephrine / metabolism*
  • Propranolol / pharmacology
  • Rats
  • Rats, Wistar
  • Stereoisomerism

Substances

  • Biogenic Monoamines
  • Propranolol
  • Droxidopa
  • Norepinephrine