Expression of core binding factor alpha1 up-regulated by IGF-I, GM-CSF, and EGF through MAPK pathway in MC3T3-E1 and C2C12 cells

Acta Pharmacol Sin. 2003 Oct;24(10):975-84.

Abstract

Aim: To study the regulating function and mechanism of insulin-like growth factor-I (IGF-I), granulocyte-macrophage colony-stimulating factor (GM-CSF), and epidermal growth factor (EGF) on murine core binding factor alpha1 (Cbfalpha1) gene expression.

Methods: Luciferase reporter gene method and RT-PCR technique were used to examine the effects of these growth factors on the promoter activity and mRNA expression of Cbfalpha1 gene in MC3T3-E1 and C2C12 cells.

Results: IGF-I (from 1 nmol/L to 1 micromol/L), GM-CSF (100 nmol/L), and EGF (1 micromol/L) increased the luciferase expression in MC3T3-E1 cells (P<0.05). And mitogen-activated protein kinase (MAPK) inhibitor, PD 98059 (10 micromol/L), completely blocked IGF-1, GM-CSF, and EGF-induced expression of Cbfa1 promoter activity (P<0.01). In C2C12 cells, IGF-I (from 1 nmol/L to 10 micromol/L), GM-CSF (100 nmol/L and 1 micromol/L), and EGF (100 nmol/L) enhanced the expression of luciferase reporter plasmid driven by mCbfalpha1 promoter (P<0.05). Addition of PD 98059 also blocked the stimulatory effects of these growth factors on Cbfalpha1 promoter activity (P<0.01). Moreover, Cbfalpha1 mRNA expression was significantly increased after treatment with IGF-I (1 nmol/L, 100 nmol/L), GM-CSF (100 nmol/L, 1 micromol/L), and EGF (1 micromol/L, 100 nmol/L) in MC3T3-E1 and C2C12 cells, respectively (P<0.05). These stimulatory effects of IGF-I, GM-CSF, and EGF on Cbfalpha1 mRNA expression were abolished by PD 98059.

Conclusion: IGF-I, GM-CSF, and EGF could increase the promoter activity and the mRNA expression of murine Cbfalpha1 gene in MC3T3-E1 and C2C12 cells. These stimulatory effects might be mediated by activating the intracellular MAPK-dependent signaling pathway.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Line
  • Core Binding Factor alpha Subunits
  • DNA-Binding Proteins / biosynthesis*
  • DNA-Binding Proteins / genetics
  • Epidermal Growth Factor / pharmacology*
  • Flavonoids / pharmacology
  • Granulocyte-Macrophage Colony-Stimulating Factor / pharmacology*
  • Insulin-Like Growth Factor I / pharmacology*
  • MAP Kinase Signaling System*
  • Mice
  • Mitogen-Activated Protein Kinases / antagonists & inhibitors
  • Myoblasts / cytology
  • Myoblasts / metabolism
  • Osteoblasts / cytology
  • Osteoblasts / metabolism
  • RNA, Messenger / genetics
  • Transcription Factors / biosynthesis*
  • Transcription Factors / genetics
  • Up-Regulation

Substances

  • Core Binding Factor alpha Subunits
  • DNA-Binding Proteins
  • Flavonoids
  • RNA, Messenger
  • Transcription Factors
  • core binding factor alpha
  • Epidermal Growth Factor
  • Insulin-Like Growth Factor I
  • Granulocyte-Macrophage Colony-Stimulating Factor
  • Mitogen-Activated Protein Kinases
  • 2-(2-amino-3-methoxyphenyl)-4H-1-benzopyran-4-one