Induction of APOBEC3G ubiquitination and degradation by an HIV-1 Vif-Cul5-SCF complex

Science. 2003 Nov 7;302(5647):1056-60. doi: 10.1126/science.1089591. Epub 2003 Oct 16.

Abstract

Human immunodeficiency virus-1 (HIV-1) Vif is essential for viral evasion of host antiviral factor CEM15/APOBEC3G. We report that Vif interacts with cellular proteins Cul5, elongins B and C, and Rbx1 to form an Skp1-cullin-F-box (SCF)-like complex. The ability of Vif to suppress antiviral activity of APOBEC3G was specifically dependent on Cul5-SCF function, allowing Vif to interact with APOBEC3G and induce its ubiquitination and degradation. A Vif mutant that interacted with APOBEC3G but not with Cul5-SCF was functionally inactive. The Cul5-SCF was also required for Vif function in distantly related simian immunodeficiency virus mac. These results indicate that the conserved Cul5-SCF pathway used by Vif is a potential target for antiviral development.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • APOBEC-3G Deaminase
  • Animals
  • Carrier Proteins / genetics
  • Carrier Proteins / metabolism
  • Cell Line
  • Cullin Proteins / genetics
  • Cullin Proteins / metabolism*
  • Cytidine Deaminase
  • Elongin
  • Gene Products, vif / genetics
  • Gene Products, vif / metabolism*
  • HIV-1 / genetics
  • HIV-1 / physiology*
  • Humans
  • Mutation
  • Nucleoside Deaminases
  • Proteins / metabolism*
  • Repressor Proteins
  • Transcription Factors / genetics
  • Transcription Factors / metabolism
  • Transfection
  • Ubiquitin / metabolism*
  • Virus Replication
  • vif Gene Products, Human Immunodeficiency Virus

Substances

  • Carrier Proteins
  • Cullin Proteins
  • Elongin
  • Gene Products, vif
  • Proteins
  • RBX1 protein, human
  • Repressor Proteins
  • Transcription Factors
  • Ubiquitin
  • vif Gene Products, Human Immunodeficiency Virus
  • Nucleoside Deaminases
  • APOBEC-3G Deaminase
  • APOBEC3G protein, human
  • Cytidine Deaminase