Molecular movement of the voltage sensor in a K channel

J Gen Physiol. 2003 Dec;122(6):741-8. doi: 10.1085/jgp.200308927. Epub 2003 Nov 10.

Abstract

The X-ray crystallographic structure of KvAP, a voltage-gated bacterial K channel, was recently published. However, the position and the molecular movement of the voltage sensor, S4, are still controversial. For example, in the crystallographic structure, S4 is located far away (>30 A) from the pore domain, whereas electrostatic experiments have suggested that S4 is located close (<8 A) to the pore domain in open channels. To test the proposed location and motion of S4 relative to the pore domain, we induced disulphide bonds between pairs of introduced cysteines: one in S4 and one in the pore domain. Several residues in S4 formed a state-dependent disulphide bond with a residue in the pore domain. Our data suggest that S4 is located close to the pore domain in a neighboring subunit. Our data also place constraints on possible models for S4 movement and are not compatible with a recently proposed KvAP model.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Female
  • Ion Channel Gating / drug effects
  • Ion Channel Gating / physiology
  • Molecular Sequence Data
  • Mutation
  • Oocytes
  • Phenanthrolines / pharmacology
  • Potassium Channels / chemistry
  • Potassium Channels / genetics
  • Potassium Channels / metabolism
  • Potassium Channels, Voltage-Gated / chemistry*
  • Potassium Channels, Voltage-Gated / genetics
  • Potassium Channels, Voltage-Gated / metabolism*
  • Potassium Channels, Voltage-Gated / physiology*
  • Protein Structure, Secondary / genetics
  • Shaker Superfamily of Potassium Channels
  • Xenopus laevis

Substances

  • Phenanthrolines
  • Potassium Channels
  • Potassium Channels, Voltage-Gated
  • Shaker Superfamily of Potassium Channels