Effect of Terplex/VEGF-165 gene therapy on left ventricular function and structure following myocardial infarction. VEGF gene therapy for myocardial infarction

J Control Release. 2003 Dec 5;93(2):175-81. doi: 10.1016/j.jconrel.2003.06.002.

Abstract

Background: We used a novel lipopolymeric gene delivery system, TeplexDNA, to transfect myocardium with plasmid vascular endothelial growth factor-165 (pVEGF) and evaluated the ability of pVEGF to preserve left ventricular function and structure after coronary ligation in a rabbit model.

Methods: New Zealand white rabbits underwent circumflex coronary ligation after direct intramyocardial injection of either Terplex alone or Terplex + 50 microg pVEGF-165. Serial echocardiography and histologic studies were performed (n = 12/group). Mortality did not differ between groups. The data is reported as the mean +/- standard deviation.

Results: Over the 21 days following coronary ligation, pVEGF-165-treated animals demonstrated significant improvement in fractional shortening (20-25%, p = 0.02), long axis two-dimensional ejection fraction (42-51%, p=0.02) and short axis m-mode ejection fraction (46-54%, p = 0.02). No significant improvements were noted in the control group. VEGF-treated animals had a 50% increase in peri-infarct vessel density and a trend towards a smaller infarct size (20% vs. 29%, p = 0.10). In animals receiving pVEGF-165, the diastolic ventricular area increased from 1.87 +/- 0.24 cm2 prior to ligation to 2.19 +/- 0.23 cm2 at 21 days following ligation, compared to an increase from 1.84 +/- 0.38 to 2.54 +/- 0.55 cm2 over the same period in control animals (p = 0.03). Similarly, the systolic ventricular area in VEGF-165 animals increased from 1.06 +/- 0.26 cm2 prior to ligation to 1.50 +/- 0.29 cm2 at 21 days following ligation, compared to an increase from 1.16 +/- 0.30 to 1.86 +/- 0.43 cm2 over the same period in the control animals (p = 0.04).

Conclusion: TerplexDNA mediated delivery of plasmid VEGF administered at the time of coronary occlusion improves left ventricular function and reduces left ventricular dilation following myocardial infarction.

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Coronary Disease / complications
  • Coronary Disease / drug therapy
  • Coronary Disease / physiopathology
  • Coronary Vessels / injuries
  • Coronary Vessels / physiopathology
  • DNA / administration & dosage
  • DNA / genetics*
  • DNA / pharmacokinetics
  • Drug Evaluation, Preclinical
  • Echocardiography
  • Genetic Therapy / methods*
  • Genetic Vectors / administration & dosage
  • Genetic Vectors / pharmacokinetics
  • Heart Ventricles / anatomy & histology
  • Heart Ventricles / drug effects*
  • Lipids / administration & dosage
  • Lipids / chemistry
  • Lipids / pharmacokinetics
  • Lipoproteins, LDL / administration & dosage
  • Lipoproteins, LDL / genetics
  • Lipoproteins, LDL / pharmacokinetics
  • Myocardial Infarction / mortality
  • Myocardial Infarction / physiopathology
  • Myocardial Infarction / therapy*
  • Plasmids / administration & dosage
  • Plasmids / genetics
  • Plasmids / pharmacokinetics
  • Polylysine / administration & dosage
  • Polylysine / genetics
  • Polylysine / pharmacokinetics
  • Polymers / administration & dosage
  • Polymers / chemistry
  • Polymers / pharmacokinetics
  • Rabbits
  • Stearates / administration & dosage
  • Stearates / pharmacokinetics
  • Stroke Volume / drug effects
  • Stroke Volume / physiology
  • Time Factors
  • Vascular Endothelial Growth Factor A / administration & dosage
  • Vascular Endothelial Growth Factor A / genetics*
  • Vascular Endothelial Growth Factor A / pharmacokinetics
  • Vascular Endothelial Growth Factors / administration & dosage
  • Vascular Endothelial Growth Factors / genetics*
  • Vascular Endothelial Growth Factors / pharmacokinetics*
  • Ventricular Function
  • Ventricular Function, Left / drug effects
  • Ventricular Function, Left / physiology

Substances

  • Lipids
  • Lipoproteins, LDL
  • Polymers
  • Stearates
  • VEGFA protein, human
  • Vascular Endothelial Growth Factor A
  • Vascular Endothelial Growth Factors
  • stearyl-poly(lysine)
  • Polylysine
  • DNA