TGF-beta-induced RhoA and p160ROCK activation is involved in the inhibition of Cdc25A with resultant cell-cycle arrest

Proc Natl Acad Sci U S A. 2003 Dec 23;100(26):15548-53. doi: 10.1073/pnas.2536483100. Epub 2003 Dec 1.

Abstract

The ability of the transforming growth factor beta (TGF-beta) signaling pathways to inhibit proliferation of most cells while stimulating proliferation of others remains a conundrum. In this article, we report that the absence of RhoA and p160ROCK activity in fibroblastic NIH 3T3 cells and its presence in epithelial NMuMG cells can at least partially explain the difference in the TGF-beta growth response. Further, evidence is presented for TGF-beta-stimulated p160ROCK translocation to the nucleus and inhibitory phosphorylation of the cyclin-dependent kinase-activating phosphatase, Cdc25A. The resultant suppression of Cdk2 activity contributes to G1/S inhibition in NMuMG cells. These data provide evidence that signaling through RhoA and p160ROCK is important in TGF-beta inhibition of cell proliferation and links signaling components for epithelial transdifferentiation with regulation of cell-cycle progression.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 3T3 Cells
  • Animals
  • Cell Cycle / drug effects
  • Cell Cycle / physiology*
  • Cell Division
  • Cell Line
  • Epithelial Cells / cytology
  • Female
  • Intracellular Signaling Peptides and Proteins
  • Mammary Glands, Animal / cytology
  • Mice
  • Phosphorylation
  • Protein Serine-Threonine Kinases / metabolism*
  • Transforming Growth Factor beta / pharmacology*
  • cdc25 Phosphatases / antagonists & inhibitors*
  • cdc25 Phosphatases / metabolism
  • rho-Associated Kinases
  • rhoA GTP-Binding Protein / metabolism*

Substances

  • Intracellular Signaling Peptides and Proteins
  • Transforming Growth Factor beta
  • Protein Serine-Threonine Kinases
  • rho-Associated Kinases
  • Cdc25a protein, mouse
  • cdc25 Phosphatases
  • rhoA GTP-Binding Protein