CCAAT/enhancer binding protein homologous protein (DDIT3) induces osteoblastic cell differentiation

Endocrinology. 2004 Apr;145(4):1952-60. doi: 10.1210/en.2003-0868. Epub 2003 Dec 18.

Abstract

CCAAT/enhancer binding protein (C/EBP) homologous protein (CHOP/DDIT3), a member of the C/EBP family of transcription factors, plays a role in cell survival and differentiation. CHOP/DDIT3 binds to C/EBPs to form heterodimers that do not bind to consensus Cebp sequences, acting as a dominant-negative inhibitor. CHOP/DDIT3 blocks adipogenesis, and we postulated it could induce osteoblastogenesis. We investigated the effects of constitutive CHOP/DDIT3 overexpression in murine ST-2 stromal cells transduced with retroviral vectors. ST-2 cells differentiated toward osteoblasts, and CHOP/DDIT3 accelerated and enhanced the appearance of mineralized nodules, and the expression of osteocalcin and alkaline phosphatase mRNAs, particularly in the presence of bone morphogenetic protein-2. CHOP/DDIT3 overexpression opposed adipogenesis, and did not cause substantial changes in cell number. CHOP/DDIT3 overexpression did not modify C/EBPalpha or -beta mRNA levels but decreased C/EBPdelta after 24 d of culture. Electrophoretic mobility shift and supershift assays demonstrated that overexpression of CHOP/DDIT3 decreased the binding of C/EBPs to their consensus sequence by interacting with C/EBPalpha and -beta, confirming its dominant-negative role. In addition, CHOP/DDIT3 enhanced bone morphogenetic protein-2/Smad signaling. In conclusion, CHOP/DDIT3 enhances osteoblastic differentiation of stromal cells, in part by interacting with C/EBPalpha and -beta and also by enhancing Smad signaling.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Alkaline Phosphatase / metabolism
  • Animals
  • Bone Morphogenetic Protein 2
  • Bone Morphogenetic Proteins / pharmacology
  • CCAAT-Enhancer-Binding Proteins / genetics
  • CCAAT-Enhancer-Binding Proteins / metabolism
  • CCAAT-Enhancer-Binding Proteins / pharmacology*
  • Cell Differentiation / drug effects
  • Cell Line
  • Drug Synergism
  • Mice
  • Osteoblasts / cytology*
  • Osteoblasts / metabolism
  • Osteoblasts / physiology
  • Osteocalcin / metabolism
  • Phenotype
  • Protein Isoforms / metabolism
  • Stromal Cells / cytology
  • Transcription Factor CHOP
  • Transcription Factors / genetics
  • Transcription Factors / pharmacology*
  • Transduction, Genetic
  • Transforming Growth Factor beta*

Substances

  • Bmp2 protein, mouse
  • Bone Morphogenetic Protein 2
  • Bone Morphogenetic Proteins
  • CCAAT-Enhancer-Binding Proteins
  • Ddit3 protein, mouse
  • Protein Isoforms
  • Transcription Factors
  • Transforming Growth Factor beta
  • Osteocalcin
  • Transcription Factor CHOP
  • Alkaline Phosphatase