Inhibition of spliceosome assembly by the cell cycle-regulated protein kinase MELK and involvement of splicing factor NIPP1

J Biol Chem. 2004 Mar 5;279(10):8642-7. doi: 10.1074/jbc.M311466200. Epub 2003 Dec 29.

Abstract

NIPP1 is a ubiquitous nuclear protein that is required for spliceosome assembly. We report here that the phosphothreonine-binding Forkhead-associated domain of NIPP1 interacts with the cell cycle-regulated protein Ser/Thr kinase MELK (maternal embryonic leucine zipper kinase). The NIPP1-MELK interaction was critically dependent on the phosphorylaton of Thr-478 of MELK and was increased in lysates from mitotically arrested cells. Recombinant MELK was a potent inhibitor of an early step of spliceosome assembly in nuclear extracts. This splicing defect was also seen with a kinase-dead mutant but was absent after mutation (T478A) of the NIPP1 binding site of MELK, indicating a mediatory role for NIPP1. Our data suggest that MELK has a role in the cell cycle-regulated control of pre-mRNA splicing.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • COS Cells
  • Carrier Proteins / metabolism*
  • Cell Cycle / physiology
  • Endoribonucleases*
  • HeLa Cells
  • Humans
  • Intracellular Signaling Peptides and Proteins*
  • Phosphoprotein Phosphatases
  • Phosphorylation
  • Protein Serine-Threonine Kinases / metabolism*
  • RNA Precursors / physiology
  • RNA Splicing
  • RNA-Binding Proteins*
  • Spliceosomes / physiology*

Substances

  • Carrier Proteins
  • Intracellular Signaling Peptides and Proteins
  • RNA Precursors
  • RNA-Binding Proteins
  • protein phosphatase inhibitor-1
  • Melk protein, mouse
  • Protein Serine-Threonine Kinases
  • Endoribonucleases
  • Phosphoprotein Phosphatases
  • PPP1R8 protein, human