Inhibitory effect of tea polyphenols on transforming growth factor-beta1 expression in rat with cyclosporine A-induced chronic nephrotoxicity

Acta Pharmacol Sin. 2004 Jan;25(1):98-103.

Abstract

Aim: To investigate the inhibitory effect of tea polyphenols (TP) on the transforming growth factor-beta1 (TGF-beta1) expression in rat model of cyclosporine A (CsA)-induced chronic nephrotoxicity.

Methods: The rat model of CsA-induced chronic nephrotoxicity was used, 4 groups of rats were respectively treated with vehicle (0.1 mL/kg/d sc), TP (80 mg/kg/d ig), CsA (15 mg/kg/d sc) and TP plus CsA (CsA 15 mg/kg/d sc+TP 80 mg/kg/d, ig). At the end of day 28 of treatment, serum and urine are analyzed for creatinine clearance, kidney tissue for pathologic analysis. The TGF-beta1 mRNA and its protein expression were detected by RT-PCR, immunohistochemistry, and Western blot.

Results: CsA-treated rats had increased renal expression of TGF-beta1 mRNA and its protein, compared with the vehicle- or TP-treated controls. The renal function and interstitial fibrosis were ameliorated and renal expression of TGF-beta1 mRNA and its protein was decreased in animals treated with CsA plus TP, compared with animals treated with CsA alone (P<0.05).

Conclusion: TP significantly inhibits renal expression of TGF-beta1 in rat model of cyclosporine-induced chronic nephrotoxicity, suggesting that the decreased renal expression of TGF-beta1 exerted by TP is one of mechanisms to protect renal function and tissue structure.

MeSH terms

  • Animals
  • Antioxidants / pharmacology
  • Cyclosporine
  • Flavonoids / isolation & purification
  • Flavonoids / pharmacology*
  • Gene Expression
  • Kidney / metabolism*
  • Kidney Diseases / chemically induced
  • Kidney Diseases / metabolism*
  • Male
  • Phenols / isolation & purification
  • Phenols / pharmacology*
  • Polyphenols
  • RNA, Messenger / genetics
  • Rats
  • Rats, Sprague-Dawley
  • Tea* / chemistry
  • Transforming Growth Factor beta / biosynthesis*
  • Transforming Growth Factor beta / genetics
  • Transforming Growth Factor beta1

Substances

  • Antioxidants
  • Flavonoids
  • Phenols
  • Polyphenols
  • RNA, Messenger
  • Tea
  • Tgfb1 protein, rat
  • Transforming Growth Factor beta
  • Transforming Growth Factor beta1
  • Cyclosporine