Susceptibility of African isolates of Plasmodium falciparum to artemisinin (qinghaosu)

Trop Med Parasitol. 1992 Sep;43(3):197-8.

Abstract

We studied in vitro susceptibility of 79 African strains of Plasmodium falciparum to artemisinin, chloroquine, quinine, mefloquine and halofantrine and the potential cross-resistance among the drugs. Most strains presented an 50% inhibitory concentration (IC50) of artemisinin below 26 nmol/liter. A positive correlation between IC50S of artemisinin and those of quinine, mefloquine and halofantrine was observed. Cross resistance between artemisinin and other antimalarials may limit its use as a replacement drug.

MeSH terms

  • Animals
  • Antimalarials / pharmacology*
  • Artemisinins*
  • Drug Resistance
  • Drugs, Chinese Herbal / pharmacology*
  • Plasmodium falciparum / drug effects*
  • Sesquiterpenes / pharmacology*

Substances

  • Antimalarials
  • Artemisinins
  • Drugs, Chinese Herbal
  • Sesquiterpenes
  • artemisinin