Genetic and phenotypic characterization of pyrazinamide-resistant mycobacterium tuberculosis complex isolates in Japan

Diagn Microbiol Infect Dis. 2004 Feb;48(2):111-6. doi: 10.1016/j.diagmicrobio.2003.09.013.

Abstract

The pncA gene mutations associated with pyrazinamide (PZA) resistance in Mycobacterium tuberculosis complex were determined in 26 PZA-resistant isolates in Japan. Of the 26 PZA-resistant isolates included, 21 were negative for pyrazinamidase (PZase). Of these, 20 isolates had various pncA mutations, resulting in alteration of primary amino acid sequence. However, 1 PZase-negative isolate did not have any mutation on pncA gene. The remaining 5 PZA-resistant isolates were positive for PZase and had identical pncA alleles with PZA-susceptible isolates. IS6110 RFLP analysis demonstrated various distinct IS6110 types and 5 pairs of isolates were very close to each other (>90% identical pattern). This study demonstrates that most of the PZA resistance is a result of various mutations on pncA resulting in loss of PZase activity. Further investigation, particularly on PZase-positive but PZA-resistant isolates and a PZase-negative isolate with no mutation on pncA, should be urgently done.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amidohydrolases / genetics*
  • Amidohydrolases / metabolism
  • Antitubercular Agents / pharmacology*
  • DNA Fingerprinting
  • DNA Transposable Elements / genetics
  • DNA, Bacterial / chemistry
  • DNA, Bacterial / genetics
  • Drug Resistance, Bacterial
  • Humans
  • Japan
  • Mutation
  • Mycobacterium tuberculosis / drug effects*
  • Mycobacterium tuberculosis / enzymology
  • Mycobacterium tuberculosis / genetics*
  • Polymerase Chain Reaction
  • Polymorphism, Restriction Fragment Length
  • Pyrazinamide / pharmacology*
  • Tuberculosis / microbiology*

Substances

  • Antitubercular Agents
  • DNA Transposable Elements
  • DNA, Bacterial
  • Pyrazinamide
  • Amidohydrolases
  • pyrazinamide deamidase