[99mTc]diphosphonate uptake and hemodynamics in experimental arthritis: effect of naproxen in the canine carrageenan injection model

J Orthop Res. 1992 Sep;10(5):647-56. doi: 10.1002/jor.1100100507.

Abstract

The impact of naproxen treatment on juxta-articular hemodynamics and bone metabolism in experimental juvenile arthritis was studied in the articular carrageenan injection model. Unilateral gonarthritis was induced for 12 weeks in eight dogs receiving naproxen (dosage, 2 mg/kg) and eight controls. Regional blood flow was assessed by the microsphere method, plasma volume by the distribution space of [125I]fibrinogen, and bone metabolism by the 2-h uptake of [99mTc]diphosphonate ([99mTc]DPD). Synovial effusion was less prominent with naproxen treatment as judged by joint fluid volume and pressure. Naproxen reduced the arthritic capsular hyperemia, almost normalized a severe blood flow increase in patella and both juxta-articular epiphyses, ameliorated an expansion of plasma volume in the patella and the distal femoral epiphysis, and normalized an increased [99mTc]DPD uptake in subchondral femoral bone and the tibial cortex. Significantly increased arteriovenous shunting in the arthritic extremity was unaffected by naproxen. The study suggests that long-term cyclooxygenase inhibition offers protection against hemodynamic and metabolic changes in juxta-articular bone secondary to synovial inflammation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Arthritis / chemically induced*
  • Arthritis / drug therapy
  • Arthritis / metabolism*
  • Bone and Bones / blood supply
  • Bone and Bones / metabolism
  • Bone and Bones / physiology
  • Capillary Permeability / physiology
  • Carrageenan / administration & dosage
  • Carrageenan / adverse effects*
  • Diphosphonates / pharmacokinetics*
  • Disease Models, Animal
  • Dogs
  • Growth Plate / blood supply
  • Growth Plate / physiology
  • Hemodynamics / drug effects
  • Homeostasis
  • Injections
  • Microspheres
  • Naproxen / pharmacology*
  • Naproxen / therapeutic use
  • Regional Blood Flow
  • Technetium / pharmacokinetics*
  • Technetium Compounds*

Substances

  • Diphosphonates
  • Technetium Compounds
  • Naproxen
  • Technetium
  • technetium Tc 99m diphosphonate
  • Carrageenan