Mechanical and thermal anti-nociception in rats after systemic administration of verapamil

Neurosci Lett. 2004 Apr 22;360(1-2):57-60. doi: 10.1016/j.neulet.2004.02.049.

Abstract

Voltage-gated Ca(2+) channels expressed in neurons may contribute to nociceptive information processing. However, the role of L-type Ca(2+) channels in pain transmission is not well understood. In this study, we examined the effects of systemically administered verapamil, an antihypertensive agent and L-type Ca(2+) channel blocker, on mechanical and thermal withdrawal thresholds in rats. Intraperitoneal injections of verapamil induced dose-dependent (3-18 mg/kg) mechanical and thermal anti-nociception in adult rats without altering their sensorimotor abilities. Our data suggest that L-type Ca(2+) channels contribute to acute nociceptive signaling and that anti-nociceptive effects may result from the blockade of these channels.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Analgesics / pharmacology*
  • Animals
  • Calcium Channels, L-Type / physiology
  • Dose-Response Relationship, Drug
  • Female
  • Hot Temperature / adverse effects*
  • Pain Measurement / drug effects*
  • Pain Measurement / methods
  • Rats
  • Rats, Sprague-Dawley
  • Touch*
  • Verapamil / pharmacology*

Substances

  • Analgesics
  • Calcium Channels, L-Type
  • Verapamil