[Effects of pentylenetetrazol at subconvulsant and convulsant dose on NMDA receptor subunits in rats]

Zhejiang Da Xue Xue Bao Yi Xue Ban. 2004 May;33(3):213-5, 224. doi: 10.3785/j.issn.1008-9292.2004.03.008.
[Article in Chinese]

Abstract

Objective: To investigate the expression of N-methyl-D-asparate (NMDA) receptor subunit proteins after administration of different doses of pentylenetetrazol (PTZ).

Methods: After ip injection of a subconvulsant (35 mg/kg) and convulsant (50 mg/kg) dose of PTZ, the rats were decapitated at different time points. The levels of cortical NR1 NR2A and NR2B subunit proteins were detected by immunoblotting.

Result: 35 mg/kg PTZ and 50 mg/kg PTZ elicited different behavioral changes (P<0.001). The NR2A subunit in the cortex significantly increased 1 h after PTZ injection (P<0.05). For the 50 mg/kg group, both the NR2A and NR2B subunits proteins increased at 1 h in the cortex and then decreased; the protein levels returned to normal after 48 h. However, NR1 subunit had no changes.

Conclusion: The NR2 subunit is involved in PTZ-induced seizure.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cerebral Cortex / chemistry*
  • Dose-Response Relationship, Drug
  • Male
  • Pentylenetetrazole / administration & dosage*
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, N-Methyl-D-Aspartate / analysis*
  • Seizures / chemically induced*
  • Seizures / metabolism

Substances

  • NR1 NMDA receptor
  • NR2B NMDA receptor
  • Receptors, N-Methyl-D-Aspartate
  • N-methyl D-aspartate receptor subtype 2A
  • Pentylenetetrazole