Surface plasmon resonance evaluation of various aminoglycoside-RNA hairpin interactions reveals low degree of selectivity

Chembiochem. 2004 Jul 5;5(7):937-42. doi: 10.1002/cbic.200300819.

Abstract

Aminoglycoside antibiotics, which are able to selectively bind to RNA, are considered to be an important lead in RNA-targeting drug discovery. In this study, surface plasmon resonance (SPR) was employed to explore the interaction of aminoglycosides with known tobramycin-binding RNA hairpins (aptamers) and an unrelated RNA hairpin. It was established that aminoglycosides have multiple interactions with RNA hairpins. Unexpectedly, the different hairpins showed comparable affinity for a set of related aminoglycosides. The observed absence of selectivity presents an extra hurdle in the discovery of novel aminoglycosides as specific drugs that target defined RNA hairpins.

MeSH terms

  • Aminoglycosides / metabolism*
  • Anti-Bacterial Agents / metabolism*
  • Base Pairing
  • Base Sequence
  • Drug Interactions
  • Evaluation Studies as Topic
  • Molecular Sequence Data
  • Nucleic Acid Conformation
  • Pharmaceutical Preparations
  • RNA / chemistry*
  • RNA / metabolism*
  • Surface Plasmon Resonance
  • Tobramycin / chemistry
  • Tobramycin / metabolism

Substances

  • Aminoglycosides
  • Anti-Bacterial Agents
  • Pharmaceutical Preparations
  • RNA
  • Tobramycin