The effect of combined androgen ablation on the expression of alpha1A-adrenergic receptor in the human prostate

Prostate. 2004 Sep 1;60(4):310-6. doi: 10.1002/pros.20070.

Abstract

Background: This study was designed to determine whether androgen ablation (AA) affects expression of alpha1A-adrenergic receptors (AR) in the human prostate.

Methods: Concentrations of alpha1A-AR mRNA were determined in benign prostatic tissue from patients undergoing surgery after a 3-month course of combined androgen ablation (CAD) therapy with leuprolide and flutamide, and a matched group of untreated patients with clinical BPH.

Results: Mean concentration of alpha1A-AR in the AA group was 0.53 +/- 0.53 SD (range 0.026-1.55) attomol/mg. Control mean was 0.29 +/- 0.22 SD (range 0.02-0.69; P = 0.3, two tailed t-test). Tissue composition did not statistically differ between the two groups. Expression of alpha1A-AR correlated with concentration of smooth muscle myosin heavy chain (SMMHC) (r = 0.84, P = 0.001). No significant differences were observed after adjusting for SMMHC content.

Conclusions: A 3-month course of CAD does not appear to have a significant effect on alpha1A-AR mRNA expression in the human prostate.

Publication types

  • Clinical Trial

MeSH terms

  • Aged
  • Androgen Antagonists / pharmacology*
  • Antineoplastic Agents, Hormonal / pharmacology
  • Flutamide / pharmacology
  • Humans
  • Leuprolide / pharmacology
  • Male
  • Middle Aged
  • Prostatic Hyperplasia / pathology
  • Prostatic Neoplasms / drug therapy*
  • Prostatic Neoplasms / pathology
  • Prostatic Neoplasms / surgery
  • RNA, Messenger / analysis
  • Receptors, Adrenergic, alpha-1 / biosynthesis*
  • Reverse Transcriptase Polymerase Chain Reaction

Substances

  • ADRA1A protein, human
  • Androgen Antagonists
  • Antineoplastic Agents, Hormonal
  • RNA, Messenger
  • Receptors, Adrenergic, alpha-1
  • Flutamide
  • Leuprolide