A new era in the management of pulmonary arterial hypertension related to scleroderma: endothelin receptor antagonism

Ann Rheum Dis. 2004 Sep;63(9):1009-14. doi: 10.1136/ard.2003.017673.

Abstract

Evidence suggests that endothelin may have a fundamental role in scleroderma pathogenesis, including pulmonary arterial hypertension (PAH)--a leading cause of death in patients with scleroderma. Development of a new class of drug, endothelin receptor antagonists, heralds an improved outlook for patients with scleroderma and related diseases. Heightened vigilance towards early detection of PAH in scleroderma and a multidisciplinary approach to diagnosis and treatment may improve clinical outcomes for these patients.

Publication types

  • Review

MeSH terms

  • Antihypertensive Agents / therapeutic use*
  • Bosentan
  • Endothelin Receptor Antagonists*
  • Endothelins / physiology
  • Humans
  • Hypertension, Pulmonary / drug therapy*
  • Hypertension, Pulmonary / etiology
  • Scleroderma, Systemic / complications*
  • Sulfonamides / therapeutic use

Substances

  • Antihypertensive Agents
  • Endothelin Receptor Antagonists
  • Endothelins
  • Sulfonamides
  • Bosentan