Beta-adrenergic and muscarinic modulation of human embryonic stem cell-derived cardiomyocytes

Cell Physiol Biochem. 2004;14(4-6):187-96. doi: 10.1159/000080326.

Abstract

Background: Embryonic stem cells provide the most promising tool for cell replacement therapy including transplantation of human embryonic stem (hES) cell- derived cardiomyocytes in the infarcted area of the heart. Here we provide data for differentiation of cardiomyocytes from hES cells and firstly describe their hormonal modulation.

Methods: Using Micro-Electrode Arrays as a novel electrical mapping technique of beating cardiomyocyte clusters within whole hES cell aggregates, we were able to measure the field potential generation and morphology changes during hormonal modulation.

Results: We found that isoproterenol provokes, similar to the mouse ES cell system, a strong positive chronotropic effect with an EC50 of around 10(-8) M. Moreover, isoproterenol stimulated with a higher EC50 value the slow field potential amplitude, FP(slow), indicating a stimulation of Ca2+ channels in ventricular-like ES cell-derived cardiomyocytes which is shown to be clearly independent from frequency modulation. In contrast, carbachol (10 microM) produced a transient negative chronotropic effect but had no effect on FP(slow).

Conclusion: The Micro-Electrode system allows measurement of ionic channel modulation and chronotropic responsiveness in a pharmacological screening setup. Moreover, all our data indicate that cardiomyocytes derived from human embryonic stem cells exhibit a physiological response to the major hormones of the vegetative nervous system and might therefore serve as an ideal candidate for the use in cell replacement strategies.

MeSH terms

  • Adrenergic beta-Agonists / pharmacology*
  • Animals
  • Carbachol / pharmacology
  • Cell Culture Techniques
  • Cell Differentiation / drug effects
  • Cell Differentiation / physiology
  • Electrophysiology
  • Embryo, Mammalian / cytology*
  • Humans
  • Isoproterenol / pharmacology
  • Membrane Potentials / drug effects
  • Membrane Potentials / physiology
  • Mice
  • Microelectrodes
  • Muscarinic Antagonists / pharmacology*
  • Myocytes, Cardiac / cytology
  • Myocytes, Cardiac / drug effects*
  • Myocytes, Cardiac / physiology
  • Stem Cells / cytology*
  • Stem Cells / physiology

Substances

  • Adrenergic beta-Agonists
  • Muscarinic Antagonists
  • Carbachol
  • Isoproterenol