Characterization of the integrin alpha v beta 6 as a fibronectin-binding protein

J Biol Chem. 1992 Mar 25;267(9):5790-6.

Abstract

Integrins are a complex family of divalent cation-dependent cell adhesion receptors composed of one alpha and one beta subunit noncovalently bound to one another. A subset of integrins contains the alpha v subunit in association with one of several beta subunits (e.g. beta 3, beta 5, beta 1). We have recently identified a novel integrin beta subunit, beta 6, that is present in a number of epithelial cell lines. Using a polyclonal antibody raised against the carboxyl-terminal peptide of beta 6, we have now identified the integrin heterodimer, alpha v beta 6, on the surface of two human carcinoma cell lines. Using affinity chromatography of lysates from the pancreatic carcinoma cell line, FG-2, we demonstrate that alpha v beta 6 binds to fibronectin, but not to vitronectin or collagen I. In contrast, the alpha v beta 5 integrin, which is also expressed on FG-2 cells, binds exclusively to vitronectin. Immobilized collagen I does not interact with alpha v integrins, but binds beta 1-containing integrins. Both alpha v beta 6 and alpha v beta 5 are eluted from their respective immobilized ligands by a hexa-peptide containing the sequence Arg-Gly-Asp (RGD). RGD is highly effective in the presence of Ca2+, somewhat less effective in Mg2+, and virtually inactive in Mn2+. These results suggest that alpha v beta 6 functions as an RGD-dependent fibronectin receptor in FG-2 carcinoma cells. In agreement with this notion, cell adhesion assays show that FG-2 cell attachment to fibronectin is only partially inhibited by anti-beta 1 integrin antibodies, implying that other fibronectin receptors may be involved. Taken together with recent reports on the vitronectin receptor function of alpha v beta 5, our results suggest that the previously described carcinoma cell integrin, alpha v beta x (Cheresh, D. A., Smith, J. W., Cooper, H. M., and Quaranta, V. (1989) Cell 57, 59-69), is a mixture of at least two different receptors: alpha v beta 5, mediating adhesion to vitronectin, and alpha v beta 6, mediating adhesion to fibronectin.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Antigens, Neoplasm*
  • Cell Line
  • Cell Membrane / metabolism
  • Chromatography, Affinity
  • Electrophoresis, Polyacrylamide Gel
  • Fibronectins / metabolism*
  • Humans
  • Integrins / isolation & purification
  • Integrins / metabolism*
  • Kinetics
  • Lung Neoplasms
  • Macromolecular Substances
  • Molecular Sequence Data
  • Pancreatic Neoplasms
  • Receptors, Fibronectin
  • Receptors, Immunologic / isolation & purification
  • Receptors, Immunologic / metabolism*
  • Substrate Specificity

Substances

  • Antigens, Neoplasm
  • Fibronectins
  • Integrins
  • Macromolecular Substances
  • Receptors, Fibronectin
  • Receptors, Immunologic
  • integrin alphavbeta6