Insulinotropic action of glucagonlike peptide-I-(7-37) in diabetic and nondiabetic subjects

Diabetes Care. 1992 Feb;15(2):270-6. doi: 10.2337/diacare.15.2.270.

Abstract

Objective: Whether glucagonlike peptide-I-(7-37) (GLP-I-[7-37]), a naturally occurring intestinal peptide, is insulinotropic in nondiabetic and non-insulin-dependent (type II) diabetic subjects.

Research design and methods: GLP-I-(7-37) or saline placebo was infused (1-5 ng.kg-1.min-1 for 30 min) in 4 nondiabetic and 11 type II diabetic subjects in the fasting and prandial state. Glucose, insulin, and GLP-I-(7-37) levels were measured.

Results: GLP-I-(7-37) infusion resulted in a 3- to 10-fold increase in peak insulin levels and in insulin area under the curve in nondiabetic and diabetic subjects. In diabetic subjects, infusion concurrent with a standard meal eliminated the postprandial glucose excursion for 60 min after the meal. Insulin-releasing potency of GLP-I-(7-37) was attenuated at decreased glucose levels.

Conclusions: GLP-I-(7-37) has potent insulinotropic effects in nondiabetic and diabetic subjects. Whether GLP-I-(7-37) is useful as a therapeutic medication in type II diabetes requires further investigation.

Publication types

  • Clinical Trial
  • Controlled Clinical Trial
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adult
  • Aged
  • Blood Glucose / metabolism*
  • Diabetes Mellitus, Type 2 / blood*
  • Eating
  • Fasting
  • Female
  • Glucagon
  • Glucagon-Like Peptide 1
  • Glucagon-Like Peptides
  • Humans
  • Insulin / blood*
  • Kinetics
  • Male
  • Middle Aged
  • Peptide Fragments
  • Peptides / pharmacology*
  • Reference Values
  • Time Factors

Substances

  • Blood Glucose
  • Insulin
  • Peptide Fragments
  • Peptides
  • Glucagon-Like Peptides
  • Glucagon-Like Peptide 1
  • Glucagon
  • glucagon-like peptide 1 (7-37)